Lipid metabolism inhibitors
Showing 1–12 of 14 results
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Bioactive Lipids
1-Aminobenzotriazole | Cytochrome P450 inhibitor
1-Aminobenztriazole (1614-12-6) is a pan-specific cytochrome P450 inhibitor acting as a suicide substrate.1,2 Blocks omega-oxidation of arachidonic...$50.00 – $185.00 Select options -
New Products
ABX-1431 | MAGL inhibitor
ABX-1431 (1446817-84-0) is a potent (IC50 = 14 nM in vitro, 2.2 nM in human PC3 cells) and very selective (>100-fold over hABHD6, >200-fold o...$60.00 – $235.00 Select options -
Apoptosis
Baicalein | Inhibitor of protein tyrosine kinase in leukemia cells
Baicalein (491-67-8) is an inhibitor of protein tyrosine kinase in leukemia (CEM) cells. Induces cell cycle arrest and apoptosis.1 Originally repor...$40.00 – $148.00 Select options -
New Products
Bempedoic acid | ATP citrate lyase inhibitor
Bempedoic acid (738606-46-7) is an inhibitor of ATP citrate lyase (ACL) and activator of AMPK used in the treatment of hypercholesterolemia.1,2 In ...$45.00 – $125.00 Select options -
Bioactive Lipids
JNJ-1661010 | FAAH inhibitor
JNJ-1661010 (681136-29-8) is a potent and selective FAAH inhibitor. Initially forms a covalent adduct with FAAH but is slowly released, IC50 = 12 n...$80.00 – $260.00 Select options -
Bioactive Lipids
JZL-184 | MAG lipase inhibitor
JZL-184 (1101854-58-3) inhibits MAG lipase (IC50=8 nM) selectively over FAAH. Irreversible. Cell permeable. References/Citations: 1) Long et ...$62.00 – $248.00 Select options -
Bioactive Lipids
LY-2183240 | Anandamide uptake inhibitor
LY-2183240 (874902-19-9) is highly potent inhibitor of cellular anandamide uptake (IC50 = 0.27nM1, 15nM2). LY-2183240 has also been found2-4 to be ...$60.00 – $240.00 Select options -
Bioactive Lipids
Nonylbenzeneboronic acid | FAAH
Nonylbenzeneboronic acid (CAS 256383-45-6) is a potent and selective inhibitor of fatty acid amide hydrolase (FAAH, the enzyme which hydrolyzes and...$30.00 – $60.00 Select options -
New Products
NVP-231 | Ceramide kinase inhibitor
NVP-231 (362003-83-6) is a reversible inhibitor of ceramide kinase (IC50 = 12 nM).1 At 10 nM, it inhibited ceramide-1-phosphate formation by >50...$40.00 – $130.00 Select options -
Bioactive Lipids
Palmitoylethanolamide | GPR-55 agonist
Palmitoylethanolamide (544-31-0) is an endogenous cannabinoid. Weak ligand for CB1 (Ki= 23.8 μM) and CB2 (Ki = 13.9 μM) receptors. Inhibits fatty a...$60.00 – $240.00 Select options -
Bioactive Lipids
PF-622 | FAAH inhibitor
PF-622 (898235-65-9) is a potent and selective irreversible FAAH inhibitor. Covalently modifies active site-serine (IC50=33 nM). Completely selecti...$60.00 – $240.00 Select options -
Bioactive Lipids
RHC-80267 | DAG Lipase inhibitor
RHC-80267 (83654-05-1) inhibits DAG Lipase activity in a variety of cell types and tissues, including canine platelets, bovine adrenal chromaffin c...$55.00 – $220.00 Select options
