Histone acetylation

Showing all 6 results

  • Cancer

    Anacardic Acid | HAT inhibitor

    Rated 0 out of 5
    Anacardic acid (16611-84-0) is a natural product found in cashew nut oil. It is an inhibitor of the histone acetyltransferases p300 and PCAF (IC50’...
    $35.00$140.00 Select options

  • Cancer

    C-646 | HAT inhibitor

    Rated 0 out of 5
    C-646 (328968-36-1) is a potent and selective inhibitor of the histone acetyl transferase p300/CBP (Ki=400 nM ). Induces apoptosis in prostate canc...
    $80.00$320.00 Select options

  • Epigenetics

    CPTH2 | HAT inhibitor

    Rated 0 out of 5
    CPTH2 (357649-93-5) is a selective inhibitor of the histone acetyltransferase Gcn5P both in vitro and in vivo (IC50 = 0.8 mM). In vitro, the HAT in...
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  • Epigenetics

    CTPB | p300 HAT activator

    Rated 0 out of 5
    CTPB (586976-24-1) is a selective activator of p300 HAT (histone acetyltransferase) selective over PCAF (p300 CPB-associated factor).1,2 Reference...
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  • Apoptosis

    Embelin | XIAP inhibitor, Apoptosis inhibitor

    Rated 0 out of 5
    Embelin (550-24-3) inhibits the lysine acetyl transferase PCAF in vitro and in vivo (in vitro IC50=7.2 mM). Inhibits H3K9 acetylation in mouse live...
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  • Apoptosis

    Garcinol | HAT inhibitor

    Rated 0 out of 5
    Garcinol (78824-30-3) is a HAT (histone acetyltransferase) inhibitor (p300 IC50=7 μM and PCAF IC50=5 μM) both in vitro and in vivo.1 It potentiates...
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