Histone acetylation
Showing all 9 results
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Bioactive Lipids
Acetyl-Coenzyme A 3Li | Acetylation and fatty acid biosynthesis cofactor
Acetyl-CoA (75520-41-1) is an essential cofactor for cellular metabolism, being an ‘activated acetate’ that shuttles its moieties back and forth du...$65.00 – $260.00 Select options -
Cancer
Anacardic Acid | HAT inhibitor
Anacardic acid (16611-84-0) is a natural product found in cashew nut oil. It is an inhibitor of the histone acetyltransferases p300 and PCAF (IC50...$35.00 – $140.00 Select options -
Cancer
C-646 | HAT inhibitor
C-646 (328968-36-1) is a potent and selective inhibitor of the histone acetyl transferase p300/CBP (Ki=400 nM ). Induces apoptosis in prostate canc...$80.00 – $320.00 Select options -
Epigenetics
CPTH2 | HAT inhibitor
CPTH2 (357649-93-5) is a selective inhibitor of the histone acetyltransferase Gcn5P both in vitro and in vivo (IC50 = 0.8 mM). In vitro, the HAT in...$69.00 – $250.00 Select options -
Epigenetics
CTPB | p300 HAT activator
CTPB (586976-24-1) is a selective activator of p300 HAT (histone acetyltransferase) selective over PCAF (p300 CPB-associated factor).1,2 Reference...$60.00 – $240.00 Select options -
Apoptosis
Embelin | XIAP inhibitor/Apoptosis inhibitor
Embelin (550-24-3) inhibits the lysine acetyl transferase PCAF in vitro and in vivo (in vitro IC50=7.2 mM). Inhibits H3K9 acetylation in mouse live...$55.00 – $220.00 Select options -
Apoptosis
Garcinol | HAT inhibitor
Garcinol (78824-30-3) is a HAT (histone acetyltransferase) inhibitor (p300 IC50=7 μM and PCAF IC50=5 μM) both in vitro and in vivo.1 It potentiates...$70.00 – $280.00 Select options -
New Products
Remodelin | Acetyltransferase NAT10 inhibitor
Remodelin (949912-58-7) is a potent and selective inhibitor of N-acetyltransferase 10 (NAT10) which is capable of acetylating microtubules and hist...$65.00 – $280.00 Select options -
New Products
WM-1119 | HAT KAT6A inhibitor
WM-1119 is a potent and selective inhibitor of the MYST family histone acetyltransferase (HAT) KAT6A (MOZ) – IC50 = 6.3 nM.1,2 Induces cell cycle e...$60.00 – $195.00 Select options
