Adrenergic
Showing all 7 results
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Adrenergic
CL-316243 | ß3-adrenergic agonist / antiobesity
CL-316243 (151126-84-0) is a potent and selective β3-adrenergic receptor agonist. (EC50= 3 nM) Displays anti-obesity and anti-diabetic effects in m...$100.00 – $375.00 Select options -
Adrenergic
Efaroxan HCl | α2 adrenergic antagonist
Efaroxan HCl (89197-00-2) is a selective α2-adrenergic receptor antagonist1 (selectivity ratio of α2/α1 = 724)4 and imidazoline receptor antagonist...$80.00 – $320.00 Select options -
Adrenergic
Formoterol hemifumarate | ß2 adrenergic agonist
Formoterol hemifumarate (43229-80-7) is a potent, long-acting agonist specific to β2 (Ki = 7.6 nM), but not β1 (Ki > 2.6 µM), adrenergic recepto...$68.00 – $200.00 Select options -
Adrenergic
Perphenazine | Antipsychotic agent
Perphenazine (58-39-9) is a clinically useful typical antipsychotic drug. The therapeutic mode of action is not well understood but it binds to a w...$25.00 – $60.00 Select options -
Adrenergic
Phenoxybenzamine HCl | Calmodulin antagonist
Phenoxybenzamine HCl (63-92-3) binds to and inhibits calmodulin in a calcium-dependent and irreversible manner (IC50= ca. 1 μM)1. A classical irrev...$30.00 – $90.00 Select options -
Adenosine
SCH-202676 | GPCR inhibitor
SCH-202676 (70375-43-8) is a reversible inhibitor of both agonist and antagonist binding to G protein-coupled receptors (GPCRs).1 IC50's = 0.1-1.7 ...$52.00 – $208.00 Select options -
Adrenergic
Terazocin HCl | Adrenergic antagonist
Terazocin HCl (63074-08-8) is an α1- and α2B-adrenoceptor antagonist (Ki = 3.3, 0.7, 1.1, 7.7, 1510 and 78.2 nM for α1A, α1B, α1D, α2B, α2A and α2C...$50.00 – $150.00 Select options
