2-APB | TRP activator
2-APB (524-95-8) is an IP3 receptor antagonist (IC50=42 μM).1 Inhibits store-operated Ca2+ channels at high concentrations (50 μM) but stimulates a...
$25.00 – $50.00
2GBI | Hv1 channel blocker
2GBI (5418-95-1) is a selective and state-dependent blocker of voltage-gated proton channels (Hv1).1 2GBI blocks the channel by binding to the volt...
$50.00 – $100.00
A-438079 HCl | P2X7 antagonist
A-438079 (899431-18-6) is a competitive P2X7 receptor antagonist (pIC50 = 6.9).1 Displayed antinociceptive effects in a rat model of neuropathic pa...
$60.00 – $225.00
A-803467 | NaV1.8 blocker
A-803467 (944261-79-4) is a potent, selective inhibitor of the TTX-resistant voltage-gated sodium channel Nav1.8. Nav1.8 is preferentially expresse...
$67.00 – $268.00
A-967079 | TRPA1 blocker
A-967079 (1170613-55-4) is a TRPA1 antagonist. Active in rat models.1 Cell permeable
1) McGaraughty et al. (2010), TRPA...
$50.00 – $200.00
AP-18 | TRPA1 blocker
AP-18 (55224-94-7) is a TRPA1 channel blocker IC50=3.1-4.5 μM in various cell lines. Reduces cinnamaldehyde-induced nociception in vivo and blocks ...
$70.00 – $280.00