Neurotransmitters
Showing 1–12 of 54 results
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Dedifferentiation
(±) Tranylcypromine hemisulfate | Demethylase inhibitor
Tranylcypromine (13492-01-8) is an irreversible and non-selective monoamine oxidase inhibitor.1,2 It has been shown to inhibit the histone demethyl...$40.00 – $150.00 Select options -
Neurosciences
1400W | iNOS inhibitor
1400W (214358-33-5) is a potent, tight-binding, slow inhibitor of inducible nitric oxide synthase (iNOS). Highly selective for iNOS3 (Ki = 7 nM) ov...$40.00 – $145.00 Select options -
Dopamine
6,7-ADTN HBr | Dopamine D1 agonist
6,7-ADTN HBr (13575-86-5) is a broad spectrum dopamine receptor agonist.1,2 Demonstrates a marked selectivity for the human dopamine D3 receptor.3...$60.00 – $260.00 Select options -
Approved Drugs
9-Hydroxyrisperidone | Risperidone metabolite
9-Hydroxyrisperidone (144598-75-4) is a pharmacologically active metabolite of risperidone, an atypical antipsychotic agent.1 Displays high affinit...$30.00 – $110.00 Select options -
Cannabinoid
AM-404 | Anandamide transport inhibitor
AM-404 (198022-70-7) inhibits anandamide transport (IC50 = 1 μM) without inhibiting anandamide amidase or activating cannabinoid receptors.1,2 Vani...$40.00 – $160.00 Select options -
Calcium Signaling
Amlodipine | L-type Ca channel blocker
Amlodipine (88150-42-9) is an anti-hypertensive L-type calcium channel blocker, which also benefits the cardiovascular system by stimulating nitric...$30.00 – $55.00 Select options -
Bioactive Lipids
Anandamide | Endogenous cannabinoid
Anandamide (94421-68-8) is an endogenous cannabinoid receptor agonist.1-3 Ki=89 nM for CB1 and 371 nM for CB2 receptors. References/Citations 1...$35.00 – $120.00 Select options -
Approved Drugs
Apomorphine HCl | Dopamine agonist
Apomorphine (41372-20-7) is an archetypal dopamine pan-receptor agonist. Displays anti-Parkinsons activity in vivo.1 Protects against MPTP-induced ...$40.00 – $120.00 Select options -
Addiction
Aripiprazole | Dopamine receptor partial agonist
Aripiprazole (129722-2-9) is a clinically useful neuroleptic and antipsychotic agent.1 Dopamine D2 receptor antagonist and autoreceptor agonist.2 I...$40.00 – $100.00 Select options -
GPCRs
Astemizole | hERG channel blocker
Astemizole (68844-77-9) is an antagonist at the histamine H1 receptor. References/Citations 1) Richards et al. (1984), Astemizole. A review of ...$30.00 – $74.00 Select options -
Cholinergics
Benztropine mesylate | Induces remyelination of neurons
Benztropine mesylate (132-17-2) is a centrally acting M1 muscarinic acetylcholine receptor antagonist (Ki=0.59 nM, rat).1 Also inhibits the dopamin...$38.00 Select options -
Cellular Metabolism
Bithionol | Glutamate dehydrogenase inhibitor
Bithionol (97-18-7) is an antihelmintic drug with bacteriostatic and fungicidal properties. Bithionol has also been found to be an inhibitor of glu...$20.00 – $50.00 Select options
