Bromodomain inhibitor

  • BI 9564 | BRD9 bromodomain inhibitor

    BI 9564 (1883429-22-8) is a potent, selective, and cell permeable inhibitor of the BRD9 bromodomain, a subunit of the switch/sucrose nonfermentable (SWI/SNF) chromatin remodeling complex (IC50 = […]

    From $60.00
  • JQ1 (+) | BET Bromodomain inhibitor

    CAS:
    1268524-70-4
    Catalog Number:
    10-1584
    Activity:
    BET Bromodomain inhibitor
    Chemical Name:
    (6S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid 1,1-dimethylethyl ester
    Molecular Weight:
    456.99
    Molecular Formula:
    C23H25ClN4O2S
    Solubility:
    Soluble in DMSO (up to 60 mg/ml) or in Ethanol (up to 46 mg/ml).
    Physical Properties:
    White solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    RT
    Stability:
    Stable for 1 year as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 2 months.
    Shipping Code:
    RT
    From $100.00
  • JQ1 | Bromodomain inhibitor

    CAS:
    1268524-69-1
    Catalog Number:
    10-1361
    Activity:
    Bromodomain inhibitor
    Chemical Name:
    (6R,S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid 1,1-dimethylethyl ester
    Molecular Weight:
    457
    Molecular Formula:
    C23H25ClN4O2S
    Solubility:
    Soluble in DMSO (up to 9 mg/ml) or in Ethanol (up to 9 mg/ml).
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    RT
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 2 months.
    Shipping Code:
    RT
    From $65.00