Inhibitors

  • Candesartan | Angiotensin II antagonist

    CAS:
    139481-59-7
    Catalog Number:
    10-2049
    Activity:
    Angiotensin II antagonist
    Chemical Name:
    2-Ethoxy-1-[[2’-(1H-tetrazol-5-yl)[1,1’-biphenyl]-4-yl]methyl]-1H-benzimidazole-7-carboxylic acid
    Alternate Names:
    CV-11974
    Molecular Weight:
    400.45
    Molecular Formula:
    C24H20N6O3
    Solubility:
    Soluble in DMSO (up to 40 mg/ml)
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.
    Shipping Code:
    RT
    From $40.00
  • CCG-4986 | RGS4 inhibitor

    CAS:
    7134-19-2
    Catalog Number:
    10-1431
    Activity:
    RGS4 inhibitor
    Chemical Names:
    Methyl-N-[(4-chlorophenyl)sulfonyl]-4-nitrobenzenesulfinimidoate
    Molecular Weight:
    374.81
    Molecular Formula:
    C13H11ClN2O5S2
    Solubility:
    Soluble in DMSO (60 mg/ml); Ethanol (5 mg/ml with warming)
    Physical Properties:
    White solid
    Purity:
    >98% TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $60.00
  • YM-254890 | Gq inhibitor

    CAS:
    568580-02-9
    Catalog Number:
    10-1590
    Activity:
    Gq inhibitor
    Source:
    Isolated from Chromobacterium sp.
    Molecular Weight:
    960.1
    Molecular Formula:
    C46H69N7O15
    Solubility:
    Soluble in DMSO (up to 10 mg/ml)
    Physical Properties:
    White or off-white lyophilized solid
    Purity:
    95% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $65.00