Prostanoid receptors & prostaglandins

  • Grapiprant | EP4 Receptor antagonist

    CAS:
    415903-37-6
    Catalog Number:
    10-4006
    Activity:
    EP4 Receptor antagonist
    Chemical Name:
    1—[2-[4-(2-Ethyl-4,6-dimethylimidazo[4,5-c]pyridine-1-yl)phenyl]ethyl]-3-(4-methylphenyl)sulfonylurea
    Alternate Names:
    CJ-023423; ARY-007
    Molecular Weight:
    491.61
    Molecular Formula:
    C26H29N5O3S
    Solubility:
    Soluble in DMSO (up to at least 10 mg/ml)
    Physical Properties:
    Off-white solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $80.00
  • TG 4-155 | EP2 receptor antagonist

    CAS:
    1164462-05-8
    Catalog Number:
    10-1574
    Activity:
    EP2 receptor antagonist
    Chemical Name:
    (2E)-N-[2-(2-Methyl-1H-indol-1-yl)ethyl]-3-(3,4,5-trimethoxyphenyl)-2-propenamide
    Molecular Weight:
    394.47
    Molecular Formula:
    C23H26N2O4
    Solubility:
    Soluble in DMSO (up to 35 mg/ml) or in Ethanol (up to 10 mg/ml).
    Physical Properties:
    Off-white solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $50.00
  • Zileuton | 5-LO inhibitor

    CAS:
    111406-87-2
    Catalog Number:
    10-1098
    Activity:
    5-LO inhibitor
    Chemical Name:
    N-(1-Benzo[b]thien-2-ylethyl)-N-hydroxyurea
    Molecular Weight:
    236.29
    Molecular Formula:
    C11H12N2O2S
    Solubility:
    Soluble in DMSO (up to 25 mg/ml).
    Physical Properties:
    White solid
    Purity:
    >98%
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $32.00