Showing 1–12 of 1147 results
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CD45
(+/-) RK-682 | Tyrosine phopshatase inhibitor
RK-682 (150627-37-5) is a protein tyrosine phosphatase inhibitor (IC50's = 54 7mu;M for CD45, 2.0 μM for VHR; did not inhibit cdc25B) originally is...$75.00 – $295.00 Select options -
Dedifferentiation
(±) Tranylcypromine hemisulfate | Demethylase inhibitor
Tranylcypromine (13492-01-8) is an irreversible and non-selective monoamine oxidase inhibitor.1,2 It has been shown to inhibit the histone demethyl...$40.00 – $150.00 Select options -
Cancer
(R)-(+)-Etomoxir Na | Carnitine palmitoyltransferase inhibitor
Etomoxir (828934-41-4) is an irreversible inhibitor of mitochondrial carnitine palmitoyl transferase 1 (CPT1).1 It is widely used to study fatty ac...$70.00 – $270.00 Select options -
Epigenetics
(R)-PFI-2 HCl | Methyltransferase SETD7 inhibitor
(R)-PFI-2 (1627607-87-7) is a potent (IC50 = 2nM) and selective SAM-dependent inhibitor of the lysine methyltransferase SETD7.1 It alters Hippo pat...$99.00 – $375.00 Select options -
Bioactive Lipids
1-Aminobenzotriazole | Cytochrome P450 inhibitor
1-Aminobenztriazole (1614-12-6) is a pan-specific cytochrome P450 inhibitor acting as a suicide substrate.1,2 Blocks omega-oxidation of arachidonic...$50.00 – $185.00 Select options -
Cardiovascular
1-EBIO | K+ channel activator; Promotes cardiomyocyte differentiation
1-EBIO (10045-45-1) is a direct activator of small-conductance Ca2+-activated K+ channels (SK) which dose-dependently relaxes rat mesenteric vessel...$40.00 – $148.00 Select options -
ADAM
1,10-Phenanthroline HCl | Zn metalloprotease inhibitor
1,10-Phenanthroline (18851-33-7) is a high affinity chelator of divalent metal ions and may be used to inhibit zinc metalloenzymes.1 It is a poten...$20.00 – $40.00 Select options -
Bone and Connective Tissue
1,4-DPCA | Prolyl hydroxylase inhibitor
1,4-DPCA (331830-20-7) is a potent inhibitor of prolyl 4-hydroxylase (IC50=2-4 μM)1. Inhibits collagen deposition via inhibition of collagen prolin...$60.00 – $220.00 Select options -
Cancer
10058-F4 | Myc inhibitor
10058-F4 (403811-55-2) effectively disables c-Myc by inhibiting the c-Myc-Max association and function1. It prevents the growth of fibroblasts in a...$50.00 – $200.00 Select options -
Neurosciences
1400W | iNOS inhibitor
1400W (214358-33-5) is a potent, tight-binding, slow inhibitor of inducible nitric oxide synthase (iNOS). Highly selective for iNOS3 (Ki = 7 nM) ov...$40.00 – $145.00 Select options -
Angiogenesis
17-AAG | HSP90 inhibitor
17-AAG (75747-14-7) is a semi-synthetic analog of geldanamycin (Cat.# 10-1084) which is less toxic and more stable. 17-AAG selectively binds to and...$28.00 – $60.00 Select options -
Cellular Stress
17-AHA-Geldanamycin | Geldanamycin affinity chromatography ligand
17-AHA-geldanamycin is a semi-synthetic analog of geldanamycin containing a linker bearing a free NH2 functional group for conjugation. Selectively...$100.00 – $400.00 Select options
