Orphan Archives | Focus Biomolecules

AM251 | Cannabinoid CB1 antagonist

CAS:

183232-66-8

Catalog Number:

10-2007

Activity:

Cannabinoid CB1 receptor antagonist

Chemical Name:

N-(Piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide

Molecular Weight:

555.24

Molecular Formula:

C₂₂H₂₁Cl₂IN₄O

Solubility:

Soluble in DMSO (up to 50 mg/ml) or in Ethanol (up to 13 mg/ml)

Physical Properties:

Off-white solid

Purity:

98% by TLC
NMR (Conforms)

Storage Temperature:

-20°C (des.)

Stability:

Stable for 1 year as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.

Shipping Code:

RT

From $72.00
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CLP-3094 | GPR142 Antagonist

CAS:

312749-73-8

Catalog Number:

10-3382

Activity:

GPR142 Antagonist

Chemical Names:

2-{[2-(4-Chlorophenoxy)ethyl]thio}-1H-benzimidazole

Molecular Weight:

304.79

Molecular Formula:

C₁₅H₁₃ClN₂OS

Solubility:

Soluble in DMSO (up to 45 mg/ml)

Physical Properties:

Off-white solid

Purity:

98% TLC
NMR (Conforms)

Storage Temperature:

RT

Stability:

Stable for 2 years as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.

Shipping Code:

RT

From $65.00
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Diphenyleneiodonium chloride | Flavoprotein inhibitor

CAS:

4673-26-1

Catalog Number:

10-2668

Activity:

Flavoprotein inhibitor

Alternate Names:

DPI

Molecular Weight:

314.55

Molecular Formula:

C₁₂H₈I • Cl

Solubility:

Soluble in DMSO (up to 5 mg/ml with warming)

Physical Properties:

White solid

Purity:

98% by TLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.

Shipping Code:

RT

From $55.00
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DJ-V 159 | GPRC6A agonist; Stimulates insulin secretion in beta cells

CAS:

2253744-53-3

Catalog Number:

10-3582

Activity:

GPCR6A agonist; Stimulates insulin secretion in beta cells

Chemical Name:

N1,N3-Bis(4-cyano-3-(trifluoromethyl)phenyl)isophthalamide

Molecular Weight:

502.37

Molecular Formula:

C₂₄H₁₂F₆N₄O₂

Solubility:

Soluble in DMSO (up to 60 mg/ml).

Physical Properties:

Off-white solid

Purity:

98% by TLC
NMR (Conforms)

Storage Temperature:

RT

Stability:

Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.

Shipping Code:

RT

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Genistein | Genistin aglycone

CAS:

446-72-0

Catalog Number:

10-2139

Activity:

Tyrosine kinase inhibitor

Chemical Name:

5,7-Dihydroxy-3-(4-hydroxyphenyl)-4H-1-benzopyran-4-one

Alternate Names:

4’,5,7-Trihydroxyisoflavone

Molecular Weight:

270.24

Molecular Formula:

C₁₅H₁₀O₅

Solubility:

Soluble in DMSO (up to 25 mg/ml) or in Ethanol (up to 4 mg/ml)

Physical Properties:

Yellow solid

Purity:

98% by TLC
NMR (Conforms)

Storage Temperature:

-20°C

Stability:

Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 week.

Shipping Code:

RT

From $30.00
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Orphan

AM251 | Cannabinoid CB1 antagonist

CLP-3094 | GPR142 Antagonist

Diphenyleneiodonium chloride | Flavoprotein inhibitor

DJ-V 159 | GPRC6A agonist; Stimulates insulin secretion in beta cells

Genistein | Genistin aglycone

EXPLORE OTHER GPCRs

Focus Biomolecules • Plymouth Meeting, PA USA • 1-855-FOCUS21

Focus Biomolecules
Plymouth Meeting, PA USA
1-855-FOCUS21

Orphan

AM251 | Cannabinoid CB1 antagonist

CLP-3094 | GPR142 Antagonist

Diphenyleneiodonium chloride | Flavoprotein inhibitor

DJ-V 159 | GPRC6A agonist; Stimulates insulin secretion in beta cells

Genistein | Genistin aglycone

EXPLORE OTHER GPCRs

Focus Biomolecules • Plymouth Meeting, PA USA • 1-855-FOCUS21

Focus Biomolecules Plymouth Meeting, PA USA1-855-FOCUS21

Focus Biomolecules
Plymouth Meeting, PA USA
1-855-FOCUS21