AM-404 | Anandamide transport inhibitor
NMR (Conforms)
Available Options
| size : | Price | Quantity | |
|---|---|---|---|
| 10 mg | $40.00 | ||
| 50 mg | $160.00 |
AM-404 (198022-70-7) inhibits anandamide transport (IC50 = 1 μM) without inhibiting anandamide amidase or activating cannabinoid receptors.1,2 Vanilloid receptors are activated by AM-404.3 Active in vivo.1
References/Citations:
1) Calignano et al. (1997), Potentiation of anandamide hypotension by the transport inhibitor AM404; Eur. J. Pharmacol., 337 R1
2) Beltramo et al. (1997), Functional role of high-affinity anandamide transport, as revealed by selective inhibition; Science, 277 1094
3) Zygmunt et al. (2000), The anandamide inhibitor AM404 activates vanilloid receptors: Eur. J. Pharmacol. 396 39
NMR (Conforms)
Safety Data Sheet:
Product Data Sheet:
Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications. Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee
AM-404 (198022-70-7) inhibits anandamide transport (IC50 = 1 μM) without inhibiting anandamide amidase or activating cannabinoid receptors.1,2 Vanilloid receptors are activated by AM-404.3 Active in vivo.1
References/Citations:
1) Calignano et al. (1997), Potentiation of anandamide hypotension by the transport inhibitor AM404; Eur. J. Pharmacol., 337 R1
2) Beltramo et al. (1997), Functional role of high-affinity anandamide transport, as revealed by selective inhibition; Science, 277 1094
3) Zygmunt et al. (2000), The anandamide inhibitor AM404 activates vanilloid receptors: Eur. J. Pharmacol. 396 39
Related products
-
Gaboxadol HCl | GABA-A receptor agonist
From $60.00CAS:85118-33-8Catalog Number:10-1168Activity:GABA-A receptor agonistAlternate Names:THIP HClChemical Name:4,5,6,7-Tetrahydroisoxazolo[5,4-c]pyridine-3-ol hydrochlorideMolecular Weight:176.6Molecular Formula:C6H8N2O2 HClSolubility:Soluble in DMSO (up to 20 mg/ml) or in Ethanol (up to 20 mg/ml).Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 3 months.Shipping Code:RT -
HC-030031 | TRPA1 blocker
From $50.00CAS:349085-38-7Catalog Number:10-1065Activity:TRPA1 blockerChemical Name:Theophylline-7-(N-4-isopropylphenyl)acetamideMolecular Weight:355.4Molecular Formula:C18H21N5O3Solubility:Soluble in DMSO (up to 25 mg/ml).Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
BCTC | TRPV1 blocker
From $60.00CAS:393514-24-4Catalog Number:10-1086Activity:TRPV1 blockerChemical Name:4-(3-Chloro-2-pyridinyl)-N-[4-(1,1-dimethylethyl)phenyl]-1-piperazinecarboxamideMolecular Weight:372.9Molecular Formula:C20H25ClN4OSolubility:Soluble in DMSO (up to 25 mg/ml) or in Ethanol (up to 15 mg/ml).Physical Properties:Off-white solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stord at -20°C for up to 2 months.Shipping Code:RT
Calculate the molar concentration, mass or volume in a solution.
Concentration × Volume × Molecular Weight = Mass
