Benzotript | Cholecystokinin antagonist

CAS:
39544-74-6
Catalog Number:
10-4497
Activity:
Cholecystokinin antagonist
Chemical Name:
(2S)-2-[(4-Chlorobenzoyl)amino]-3-(1H-indol-3-yl)propanoic acid
Molecular Weight:
342.78
Molecular Formula:
C18H15ClN2O3
Solubility:
Soluble in DMSO (up to at least 25 mg/ml)
Physical Properties:
White solid
Purity:
98% by TLC
NMR (Conforms)
Storage Temperature:
-20°C
Stability:
Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
Shipping Code:
RT

Available Options

Size :PriceQuantity 
10 mg$50.00
50 mg$165.00

Benzotript (39544-74-6) antagonizes the interaction of cholecystokinin and related peptides with the cholecystokinin receptor.1  It has been reported to potentiate morphine analgesia via interaction with opioid receptors.2

References/Citations:

1) Hahne (1981), Proglumide and benzotript: Members of a different class of cholecystokinin receptor antagonists; Proc. Natl. Acad. Sci. USA. 78 6304
2) Gaudreau et al. (1990), Cholecystokinin antagonists proglumide, lorglumide and benzotript, but not L-364,718, interact with brain opioid binding sites; Neuropeptides 16 51

CAS:
39544-74-6
Catalog Number:
10-4497
Activity:
Cholecystokinin antagonist
Chemical Name:
(2S)-2-[(4-Chlorobenzoyl)amino]-3-(1H-indol-3-yl)propanoic acid
Molecular Weight:
342.78
Molecular Formula:
C18H15ClN2O3
Solubility:
Soluble in DMSO (up to at least 25 mg/ml)
Physical Properties:
White solid
Purity:
98% by TLC
NMR (Conforms)
Storage Temperature:
-20°C
Stability:
Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
Shipping Code:
RT

Safety Data Sheet:

N/A

Product Data Sheet:

Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications. Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee

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