GO289 | CK2 inhibitor
NMR (Conforms)
Available Options
| Size: | Price | Quantity | |
|---|---|---|---|
| 5 mg | $95.00 | ||
| 25 mg | $350.00 |
GO289 (694522-87-7) is a potent inhibitor of casein kinase 2 (CK2; IC50 = 7 nM).1 Showed no inhibition of DYRK, HIPK, CLK, and PIM family kinases. It is a circadian clock modifier that caused strong period lengthening. Growth of MLL-AF9 leukemia cells was strongly inhibited by GO289.
References/Citations:
- Oshima et al. (2019), Cell-based screen identifies a new potent and highly selective CK2 inhibitor for modulation of circadian rhythms and cancer cell growth; Sci. Adv. 5 eauu9060
NMR (Conforms)
Safety Data Sheet:
Product Data Sheet:
Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications. Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee
GO289 (694522-87-7) is a potent inhibitor of casein kinase 2 (CK2; IC50 = 7 nM).1 Showed no inhibition of DYRK, HIPK, CLK, and PIM family kinases. It is a circadian clock modifier that caused strong period lengthening. Growth of MLL-AF9 leukemia cells was strongly inhibited by GO289.
References/Citations:
- Oshima et al. (2019), Cell-based screen identifies a new potent and highly selective CK2 inhibitor for modulation of circadian rhythms and cancer cell growth; Sci. Adv. 5 eauu9060
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