H2L5186303 | LPA2 antagonist
NMR (Conforms)
Available Options
| Size : | Price | Quantity | |
|---|---|---|---|
| 5 mg | $60.00 | ||
| 25 mg | $200.00 |
H2L5186303 (139262-76-3) is a potent and selective lysophosphatidic acid 2 (LPA2) receptor antagonist. IC50 = 8.9 nM, 1230 nM and 27.35 μM for LPA2, LPA3, and LPA1 respectively.1,2
References/Citations:
1) Fells et al. (2008) Identification of non-lipid LPA3 antagonists by virtual screening; Bioorg. Med. Chem. 16 6207
2) Fells et al. (2009) Structure-based drug design identifies novel LPA3 antagonists; Bioorg. Med. Chem. 17 7457
NMR (Conforms)
Safety Data Sheet:
Product Data Sheet:
Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications. Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee
H2L5186303 (139262-76-3) is a potent and selective lysophosphatidic acid 2 (LPA2) receptor antagonist. IC50 = 8.9 nM, 1230 nM and 27.35 μM for LPA2, LPA3, and LPA1 respectively.1,2
References/Citations:
1) Fells et al. (2008) Identification of non-lipid LPA3 antagonists by virtual screening; Bioorg. Med. Chem. 16 6207
2) Fells et al. (2009) Structure-based drug design identifies novel LPA3 antagonists; Bioorg. Med. Chem. 17 7457
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