JNJ-1661010 | FAAH inhibitor
NMR (Conforms)
Available Options
| size : | Price | Quantity | |
|---|---|---|---|
| 10 mg | $80.00 | ||
| 50 mg | $260.00 |
JNJ-1661010 (681136-29-8) is a potent and selective FAAH inhibitor. Initially forms a covalent adduct with FAAH but is slowly released, IC50 = 12 nM. 100-fold selectivity for FAAH-1 over FAAH-2. Cell permeable and active in vivo. JNJ-1661010 displays analgesic activity in various animal models.
References/Citations:
1) Karbarz et al. (2009), Biochemical and biological properties of 4-(3-phenyl-[1,2,4]thiadiazol-5-yl)-piperazine-1-carboxylic acid phenylamide, a mechanism-based inhibitor of fatty acid amide hydrolase; Anesth. Analg., 108 316
NMR (Conforms)
Safety Data Sheet:
Product Data Sheet:
Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications. Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee
JNJ-1661010 (681136-29-8) is a potent and selective FAAH inhibitor. Initially forms a covalent adduct with FAAH but is slowly released, IC50 = 12 nM. 100-fold selectivity for FAAH-1 over FAAH-2. Cell permeable and active in vivo. JNJ-1661010 displays analgesic activity in various animal models.
References/Citations:
1) Karbarz et al. (2009), Biochemical and biological properties of 4-(3-phenyl-[1,2,4]thiadiazol-5-yl)-piperazine-1-carboxylic acid phenylamide, a mechanism-based inhibitor of fatty acid amide hydrolase; Anesth. Analg., 108 316
Related products
-
U-18666A | Cholesterol transport inhibitor
From $80.00CAS:3039-71-2Catalog Number:10-1075Activity:Cholesterol transport inhibitorChemical Name:3ß-[2-(Diethylamino)ethoxy]androst-5-en-17-one hydrochlorideMolecular Weight:424.07Molecular Formula:C25H41NO2·HClSolubility:Soluble in DMSO (up to 30 mg/ml) or in Water (up to 30 mg/ml).Physical Properties:White or off-white solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 1 week.Shipping Code:RT -
DCHA-Gly | Endogenous lipo-amino acid
From $50.00CAS:132850-40-9Catalog Number:10-1316Activity:Endogenous lipo-amino acidChemical Name:N-DocosahexaenoylglycineMolecular Weight:385.55Molecular Formula:C24H35NO3Solubility:Soluble in DMSO (up to 25 mg/ml) or in Ethanol (up to 25 mg/ml).Physical Properties:Yellowish waxy solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Product is prone to air oxidation. Solutions in degassed DMSO or ethanol may be stored at -20° for up to 1 month under a nitrogen/argon atmosphere.Shipping Code:RT -
NA-Gly | GPR18 agonist
From $60.00CAS:179113-91-8Catalog Number:10-1200Activity:GPR18 agonistAlternate Names:N-ArachidonylglycineChemical Name:N-(5Z,8Z,11Z,14Z-eicosatetraenoyl)glycineMolecular Weight:361.53Molecular Formula:C22H35NO3Solubility:Soluble in DMSO (up to 50 mg/ml).Physical Properties:Beige waxy solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Product is subject to oxidation. Solutions in degassed DMSO may be stored at -20°C for up to 1 month.Shipping Code:Blue Ice
Calculate the molar concentration, mass or volume in a solution.
Concentration × Volume × Molecular Weight = Mass
20% OFF
For Postdoc
Customers!
Focus Biomolecules • Plymouth Meeting, PA USA • 1-855-FOCUS21
Focus Biomolecules
Plymouth Meeting, PA USA
1-855-FOCUS21
Website Created by Advanta Advertising LLC.