K252B | Kinase inhibitor (pan-specific)
NMR (Conforms)
Available Options
| size : | Price | Quantity | |
|---|---|---|---|
| 100 µg | $60.00 | ||
| 1 mg | $275.00 |
K252B (99570-78-2) is a potent pan-specific protein kinase inhibitor: PKA (Ki = 20 nM), PKG (Ki = 100 nM)1 as well as other kinases. Cell impermeable.2
References/Citations:
1) Kase et al. (1987), K252 compounds, novel and potent inhibitors of protein kinase C and cyclic nucleotide-dependent protein kinases; Biochem. Biophys. Res. Commun., 142 436
2) Makino et al. (2012), Inhibition of uterine sarcoma cell growth through suppression of endogenous tyrosine kinase B signaling; PLoS One, 7 e41049
NMR (Conforms)
Safety Data Sheet:
Product Data Sheet:
Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications. Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee
K252B (99570-78-2) is a potent pan-specific protein kinase inhibitor: PKA (Ki = 20 nM), PKG (Ki = 100 nM)1 as well as other kinases. Cell impermeable.2
References/Citations:
1) Kase et al. (1987), K252 compounds, novel and potent inhibitors of protein kinase C and cyclic nucleotide-dependent protein kinases; Biochem. Biophys. Res. Commun., 142 436
2) Makino et al. (2012), Inhibition of uterine sarcoma cell growth through suppression of endogenous tyrosine kinase B signaling; PLoS One, 7 e41049
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