MS012 | Potent and selective GLP lysine methyltransferase inhibitor
NMR (Conforms)
Available Options
| Size: | Price | Quantity | |
|---|---|---|---|
| 5 mg | $75.00 | ||
| 25 mg | $250.00 |
MS012 (2089617-83-2) is a highly potent (IC50 = 7 nM) and selective (140-fold over the related lysine methyltransferase G9a) inhibitor of G9a-Like Protein (GLP) Lysine Methyltransferase. It was also selective for GLP over a panel of 29 other methyltransferases.
References/Citations:
- Xiong et al. (2017) Discovery of Potent and selective Inhibitors for G9a-Like Protein (GLP) Lysine Methyltransferase; J. Med.Chem. 60 1876
NMR (Conforms)
Safety Data Sheet:
Product Data Sheet:
Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications. Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee
MS012 (2089617-83-2) is a highly potent (IC50 = 7 nM) and selective (140-fold over the related lysine methyltransferase G9a) inhibitor of G9a-Like Protein (GLP) Lysine Methyltransferase. It was also selective for GLP over a panel of 29 other methyltransferases.
References/Citations:
- Xiong et al. (2017) Discovery of Potent and selective Inhibitors for G9a-Like Protein (GLP) Lysine Methyltransferase; J. Med.Chem. 60 1876
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