OX04528 | GPR84 agonist
NMR (Conforms)
Available Options
| Size: | Price | Quantity | |
|---|---|---|---|
| 5 mg | $80.00 | ||
| 25 mg | $295.00 |
OX04528 (3028055-45-7) is a very potent (cAMP EC50 = 5.98 pM), selective (inactive at GPR40, GPR120, and CB2), and orally bioavailable GPR84 agonist with no detectable effects on ß-arrestin recruitment. A potent new chemical tool to probe the role of GPR84 in cancer, inflammatory, and fibrotic diseases.
References/Citations:
- Wang et al. (2024), Development of Highly Potent, G-Protein Biased, Selective, and Orally Bioavailable GPR84 Agonists; J. Med. Chem. 67 110
NMR (Conforms)
Safety Data Sheet:
Product Data Sheet:
Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications. Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee
OX04528 (3028055-45-7) is a very potent (cAMP EC50 = 5.98 pM), selective (inactive at GPR40, GPR120, and CB2), and orally bioavailable GPR84 agonist with no detectable effects on ß-arrestin recruitment. A potent new chemical tool to probe the role of GPR84 in cancer, inflammatory, and fibrotic diseases.
References/Citations:
- Wang et al. (2024), Development of Highly Potent, G-Protein Biased, Selective, and Orally Bioavailable GPR84 Agonists; J. Med. Chem. 67 110
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