PSB-22269 | GPR17 antagonist

CAS:
 N/A
Catalog Number:
 10-4469
PSB-22269 chemical structure

Available Options

Size:PriceQuantity 
5 mg$90.00
25 mg$340.00

PSB-22269 is a potent competitive antagonist (Ki = 8.91 nM; pIC50 = 7.0) of GPR17, an orphan receptor involved in inflammatory diseases.

References/Citations:

  1. Boshta et al. (2024), Discovery of Anthranilic Acid Derivatives as Antagonists of the Pro-Inflammatory Orphan G Protein-Coupled Receptor GPR17; J. Med. Chem., 67 19365
GPR17 antagonist, PSB-22269, PSB-22269 supplier, PSB22269
CAS:
N/A
Catalog Number:
10-4469
Activity:
GPR17 antagonist
Chemical Names:
5-Methoxy-2-(5-(3’methoxy-[1,1’-biphenyl]-2-yl)furan-2-carboxamido)benzoic acid
Molecular Weight:
443.46
Molecular Formula:

C26H21NO6

Solubility:
Soluble in DMSO (100 mg/ml)
Physical Properties:
Off-white/gray solid
Purity:

>98% HPLC
NMR: (Conforms)

Storage Temperature:
-20°C
Stability:
Stable for up to 2 years when stored as supplied @ -20°C. Solutions in DMSO may be stored at -20°C for up to 3 months.
Shipping Code:
RT

Safety Data Sheet:

N/A

Product Data Sheet:

Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications. Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee