PSB-KK1445 | GPR18 agonist
Available Options
| Size: | Price | Quantity | |
|---|---|---|---|
| 5 mg | $60.00 | ||
| 25 mg | $215.00 |
PSB-KK1445 (885896-54-8) is a potent (EC50 = 45.4 nM human; 124 nM mouse) and highly selective (>200-fold over CB1, CB2, GPR55, and GPR183) GPR18 agonist. A new chemical tool to explore the role of GPR18 in cancer and immunology.
References/CItations:
- Mahardhika et al. (2024), Potent, Selective Agonists for the Cannabinoid-like Orphan G Protein-Coupled Receptor GPR18: A Promising Drug Target for Cancer and Immunity; J.Med.Chem. 67 9896
C24H23FN6O2
>98% HPLC
NMR: (Conforms)
Safety Data Sheet:
Product Data Sheet:
Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications. Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee
PSB-KK1445 (885896-54-8) is a potent (EC50 = 45.4 nM human; 124 nM mouse) and highly selective (>200-fold over CB1, CB2, GPR55, and GPR183) GPR18 agonist. A new chemical tool to explore the role of GPR18 in cancer and immunology.
References/CItations:
- Mahardhika et al. (2024), Potent, Selective Agonists for the Cannabinoid-like Orphan G Protein-Coupled Receptor GPR18: A Promising Drug Target for Cancer and Immunity; J.Med.Chem. 67 9896
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