GABAA

  • Allopregnanolone | GABA-A positive allosteric modulator

    CAS:
    516-54-1
    Catalog Number:
    10-3489
    Activity:
    GABA-A positive allosteric modulator
    Chemical Name:
    (3α,5α)-3-Hydroxy-pregnan-20-one
    Alternate Name:
    (3α,5α)-Tetrahydroprogesterone; 3-OH-DHP
    Molecular Weight:
    318.49
    Molecular Formula:
    C21H34O2
    Solubility:
    Soluble in DMSO (up to 32 mg/ml) or in Ethanol (up to 32 mg/ml)
    Physical Properties:
    White or off-white solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20° (des.)
    Stability:
    Stable for 2 years as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 1 month.
    Shipping Code:
    RT
    From $70.00
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  • Flumazenil | Benzodiazepine antagonist

    CAS:
    78755-81-4
    Catalog Number:
    10-1081
    Activity:
    Benzodiazepine antagonist
    Chemical Name:

    8-Fluoro-5,6-dihydro-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylic acid, ethyl ester

    Alternate Names:

    Ro 1722;  Ro 15-1788

    Molecular Weight:
    303.29
    Molecular Formula:
    C15H14FN3O3
    Solubility:
    Soluble in DMSO (up to 8 mg/ml)
    Physical Properties:
    White solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C (des.)
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $50.00
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  • Flupirtine maleate | K+ channel activator

    CAS:
    75507-68-5
    Catalog Number:
    10-2416
    Activity:
    K+ channel activator
    Chemical Name:
    N-[2-Amino-6-[[(4-fluorophenyl)methyl]amino]-3-pyridinyl]carbamic acid ethyl ester maleate
    Alternate Names:
    D9998
    Molecular Weight:
    420.39
    Molecular Formula:
    C15H17FN4O2 • C4H4O4
    Solubility:
    Soluble in DMSO (up to 40 mg/ml) or in Ethanol (up to 4 mg/ml)
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    RT
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $55.00
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  • Gaboxadol HCl | GABA-A receptor agonist

    CAS:
    64603-91-4
    Catalog Number:
    10-1168
    Activity:
    GABA-A receptor agonist
    Alternate Names:
    THIP HCl
    Chemical Name:
    4,5,6,7-Tetrahydroisoxazolo[5,4-c]pyridine-3-ol hydrochloride
    Molecular Weight:
    176.6
    Molecular Formula:
    C6H8N2O2 HCl
    Solubility:
    Soluble in DMSO (up to 20 mg/ml) or in Ethanol (up to 20 mg/ml).
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    RT
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $60.00
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  • Muscimol HBr | GABA-A agonist

    CAS:
    18174-72-6
    Catalog Number:
    10-1448
    Activity:
    GABA-A receptor agonist
    Chemical Name:
    5-Aminomethyl-3-hydroxyisoxazole hydrobromide
    Molecular Weight:
    234.21
    Molecular Formula:
    C14H6N2O2 •HBr
    Solubility:
    Soluble in Water (up to 10 mg/ml). Also soluble in DMSO and Ethanol.
    Physical Properties:
    White solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in distilled water may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $60.00
    View Product This product has multiple variants. The options may be chosen on the product page
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