SB-366791 | TRPV1 blocker

CAS:
472981-92-3
Catalog Number:
10-1217
Activity:
TRPV1 blocker
Chemical Name:
3-(4-Chlorophenyl)-N-(3-methoxyphenyl)-2-propenamide
Molecular Weight:
287.75
Molecular Formula:
C16H14ClNO2
Solubility:
Soluble in DMSO (up to 25 mg/ml).
Physical Properties:
White solid
Purity:
98% by TLC
NMR (Conforms)
Storage Temperature:
-20°C
Stability:
Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
Shipping Code:
RT

Available Options

size :PriceQuantity 
10 mg$60.00
50 mg$240.00

SB-366791 (472981-92-3) is a potent (IC50 = 0.7 µM) and selective TRPV1 blocker.1,2 Selective for TRPV1 in a panel of 47 different binding assays.

References/Citations:

1) Gunthorpe, et al., (2004) Identification and characterization of SB-366791, a potent and selective vanilloid receptor (VR1/TRPV1) antagonist; Neuropharmacology 46 133
2) Varga et al. (2005) Effects of the novel TRPV1 receptor antagonist SB366791 in vitro and in vivo in the rat; Neurosci. Lett.. 385 137

CAS:
472981-92-3
Catalog Number:
10-1217
Activity:
TRPV1 blocker
Chemical Name:
3-(4-Chlorophenyl)-N-(3-methoxyphenyl)-2-propenamide
Molecular Weight:
287.75
Molecular Formula:
C16H14ClNO2
Solubility:
Soluble in DMSO (up to 25 mg/ml).
Physical Properties:
White solid
Purity:
98% by TLC
NMR (Conforms)
Storage Temperature:
-20°C
Stability:
Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
Shipping Code:
RT

Safety Data Sheet:

Product Data Sheet:

Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications. Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee

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