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SR-144528 | Cannabinoid CB2 antagonist

CAS:
192703-06-3
Catalog Number:
10-1164
Activity:
Cannabinoid CB2 antagonist
Chemical Name:
5-(4-Chloro-3-methylphenyl)-1-[(4-methylphenyl)methyl]-N-[(1S,2S,4R)-1,3,3-trimethylbicyclo[2.2.1]hept-2-yl]-1H-pyrazole-3-carboxamide
Molecular Weight:
476.07
Molecular Formula:
C29H34ClN3O
Solubility:
Soluble in DMSO (up to 20 mg/ml, with warming).
Physical Properties:
Off-white solid
Purity:
98% by TLC
NMR (Conforms)
Storage Temperature:
-20°C
Stability:
Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
Shipping Code:
RT

Available Options

Size:PriceQuantity 
5 mg$100.00
25 mg$400.00

SR-144528 (192703-06-3) is a potent and selective antagonist of the cannabinoid CB2 receptor.1,2

References/Citations:

1) Rinaldi-Carmona et al. (1998), SR-144528, the first potent and selective antagonist of the CB2 cannabinoid receptor; J. Pharmacol. Exp. Ther., 284 644
2) Portier et al. (1999), SR-144528, an antagonist for the peripheral cannabinoid receptor that behaves as an inverse agonist; J. Pharmacol. Exp. Ther., 288 582

192703-06-3, Cannabinoid CB2 antagonist, SR-144528, SR-144528 supplier, SR144528
CAS:
192703-06-3
Catalog Number:
10-1164
Activity:
Cannabinoid CB2 antagonist
Chemical Name:
5-(4-Chloro-3-methylphenyl)-1-[(4-methylphenyl)methyl]-N-[(1S,2S,4R)-1,3,3-trimethylbicyclo[2.2.1]hept-2-yl]-1H-pyrazole-3-carboxamide
Molecular Weight:
476.07
Molecular Formula:
C29H34ClN3O
Solubility:
Soluble in DMSO (up to 20 mg/ml, with warming).
Physical Properties:
Off-white solid
Purity:
98% by TLC
NMR (Conforms)
Storage Temperature:
-20°C
Stability:
Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
Shipping Code:
RT

Safety Data Sheet:

Product Data Sheet:

Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications. Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee