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Astemizole | hERG channel blocker

Astemizole (68844-77-9) is an antagonist at the histamine H1 receptor.

References/Citations
1) Richards et al. (1984), Astemizole. A review of its pharmacodynamic properties and therapeutic efficacy; Drugs, 28 38
2) Laduron et al. (1982), In vitro and in vivo binding characteristics of a new long-acting histamine H1 antagonist, astemizole; Mol. Pharmacol., 21 294

Weight 1 mg
Dimensions 1 × 1 cm
Size:

10 mg, 50 mg

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CAS:
68844-77-9
Catalog Number:
10-1064
Activity:
hERG channel blocker
Chemical Name:
1-[(4-Fluorophenyl)methyl]-N-[1-[2-(4-methoxyphenyl)ethyl]-4-piperidinyl]-1H-benzimidazol-2-amine
Molecular Weight:
457.58
Molecular Formula:
C28H31FN4O
Solubility:
Soluble in DMSO (up to 25 mg/ml) or in Ethanol (up to 25 mg/ml).
Physical Properties:
White solid
Purity:
99% by TLC
NMR (Conforms)
Storage Temperature:
RT
Stability:
Stable for 1 year as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
Shipping Code:
RT

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Astemizole | hERG channel blocker

$30.00 – $74.00

CAS:
68844-77-9
Catalog Number:
10-1064
Activity:
hERG channel blocker
Chemical Name:
1-[(4-Fluorophenyl)methyl]-N-[1-[2-(4-methoxyphenyl)ethyl]-4-piperidinyl]-1H-benzimidazol-2-amine
Molecular Weight:
457.58
Molecular Formula:
C28H31FN4O
Solubility:
Soluble in DMSO (up to 25 mg/ml) or in Ethanol (up to 25 mg/ml).
Physical Properties:
White solid
Purity:
99% by TLC
NMR (Conforms)
Storage Temperature:
RT
Stability:
Stable for 1 year as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
Shipping Code:
RT
  • 10 mg
  • 50 mg
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Products Astemizole | hERG channel blocker