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Product Details

H2L5186303 | LPA2 antagonist

H2L5186303 (139262-76-3) is a potent and selective lysophosphatidic acid 2 (LPA2) receptor antagonist.  IC50 = 8.9 nM, 1230 nM and 27.35 μM for LPA2, LPA3, and LPA1 respectively.1,2

References/Citations

1) Fells et al. (2008) Identification of non-lipid LPA3 antagonists by virtual screening; Bioorg. Med. Chem. 16 6207
2) Fells et al. (2009) Structure-based drug design identifies novel LPA3 antagonists; Bioorg .Med. Chem. 17 7457

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Catalog#  10-1452

$75.00
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Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee.
 
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CAS:
139262-76-3
Catalog Number:
10-1452
Activity:
LPA2 antagonist
Chemical Name:
(Z,Z)-4,4'-[1,3-Phenylenebis(oxy-4,1-phenyleneimino)]bis[4-oxo-2-butenoic acid]
Molecular Weight:
488.45
Molecular Formula:
C26H202O8
Solubility:
Soluble in DMSO (up to 50 mg/ml).
Physical Properties:
Yellow solid
Purity:
98% by TLC
NMR (Conforms)
Storage Temperature:
-20°C
Stability:
Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
Shipping Code:
RT
Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications.

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