Nafamostat Mesylate | Serine protease inhibitor

Nafamostat mesylate (82956-11-4) is a potent and reversible serine protease inhibitor (IC50‘s range from 0.3 – 54.0 μM). Inhibits the demethylase activity of the fat mass and obesity-associated protein (FTO).1 Cell permeable. Intended for cell culture or in vivo laboratory experimentation. This product is not approved for human therapeutic use.

 

References/Citations

1) Han et al. (2019) Identification of nafamostat mesilate as an inhibitor of the fat mass and obesity-associated protein (FTO) demethylase; Chemico-Biological Interactions, 297 80

Weight 1 mg
Dimensions 1 × 1 × 1 cm
size :

10 mg, 50 mg

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CAS:
82956-11-4
Catalog Number:
10-1089
Activity:
Serine protease inhibitor
Alternate Names:
Futhan; FUT-175
Chemical Name:
6-Amidino-2-naphthyl-4-guanidinobenzoate dimesylate
Molecular Weight:
539.59
Molecular Formula:
C19H17N5O2 2CH4O3S
Solubility:
Soluble in Water (up to 25 mg/ml).
Physical Properties:
White solid
Purity:
98% by TLC
NMR (Conforms)
Storage Temperature:
RT
Stability:
Stable for 2 years as supplied. Solutions in distilled water may be stored at 4°C for up to 1 month, or at -80°C for up to 6 months.
Shipping Code:
RT

Nafamostat Mesylate | Serine protease inhibitor

$50.00$200.00

CAS:
82956-11-4
Catalog Number:
10-1089
Activity:
Serine protease inhibitor
Alternate Names:
Futhan; FUT-175
Chemical Name:
6-Amidino-2-naphthyl-4-guanidinobenzoate dimesylate
Molecular Weight:
539.59
Molecular Formula:
C19H17N5O2 2CH4O3S
Solubility:
Soluble in Water (up to 25 mg/ml).
Physical Properties:
White solid
Purity:
98% by TLC
NMR (Conforms)
Storage Temperature:
RT
Stability:
Stable for 2 years as supplied. Solutions in distilled water may be stored at 4°C for up to 1 month, or at -80°C for up to 6 months.
Shipping Code:
RT
  • 10 mg
  • 50 mg
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