AZD-2098 | CCR4 antagonist

AZD-2098 is a potent, orally bioavailable antagonist of CCR4 (pIC50 = 7.8(h), 8.0(r), 8.0(m), 7.6(d)).1 Inactive at CXCR1/2, CCR1, CCR2b, CCR5, CCR7, and CCR8 @ 10 µM.

Reference:

  1. Kindon et al. (2017), Discovery of AZD-2098 and AZD-1678, Two Potent and Bioavailable CCR4 Receptor Antagonists; ACS Med. Chem. Lett. 8 981
Weight 0.1 mg
Dimensions 0.1 × 0.1 × 0.1 cm
Size:

5 mg, 25 mg

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CAS:
566203-88-1
Catalog Number:
10-4262
Activity:
CCR4 antagonist
Chemical Names:
2,3-Dichloro-N-(3-methoxypyrazine-2-yl)benzenesulfonamide
Molecular Weight:
334.17
Molecular Formula:
C11H9Cl2N3O3S
Solubility:
Soluble in DMSO (>25 mg/ml)
Physical Properties:
Off-white/beige solid
Purity:
>98% HPLC
NMR (Conforms)
Storage Temperature:
-20°C
Stability:
Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
Shipping Code:
RT

AZD-2098 | CCR4 antagonist

$50.00$185.00

CAS:
566203-88-1
Catalog Number:
10-4262
Activity:
CCR4 antagonist
Chemical Names:
2,3-Dichloro-N-(3-methoxypyrazine-2-yl)benzenesulfonamide
Molecular Weight:
334.17
Molecular Formula:
C11H9Cl2N3O3S
Solubility:
Soluble in DMSO (>25 mg/ml)
Physical Properties:
Off-white/beige solid
Purity:
>98% HPLC
NMR (Conforms)
Storage Temperature:
-20°C
Stability:
Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
Shipping Code:
RT
  • 5 mg
  • 25 mg
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Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications.

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