PBA | TRPM4 channel blocker
Available Options
| Size: | Price | Quantity | |
|---|---|---|---|
| 5 mg | $80.00 | ||
| 25 mg | $275.00 |
PBA (3128041-29-9) is a potent and selective TRPM4 channel blocker (IC50(HCT116) = 0.15 µM; IC50(HEK293) = 0.34 µM). Active in both human and mouse. TRPM4 blockers are of interest in treating cardiovascular diseases, neuronal diseases, and cancer
References/Citations:
- Gerber et al. (2026), Potent Anthranillic Anilide-Based TRPM4 Channel Inhibitors Identified by a Structure-Activity Relationship Study; J. Med. Chem. 69 8763
Safety Data Sheet:
Product Data Sheet:
Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications. Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee
PBA (3128041-29-9) is a potent and selective TRPM4 channel blocker (IC50(HCT116) = 0.15 µM; IC50(HEK293) = 0.34 µM). Active in both human and mouse. TRPM4 blockers are of interest in treating cardiovascular diseases, neuronal diseases, and cancer
References/Citations:
- Gerber et al. (2026), Potent Anthranillic Anilide-Based TRPM4 Channel Inhibitors Identified by a Structure-Activity Relationship Study; J. Med. Chem. 69 8763
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