PARP
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Olaparib | PARP1 inhibitor
From $45.00CAS:763113-22-0Catalog Number:10-2154Activity:PARP1 inhibitorChemical Name:4-(3-(4-(Cyclopropanecarbonyl)piperazine-1-carbonyl)-4-fluorobenzyl)phthalazine-1(2H)-oneAlternate Names:AZD-2281; KU-59436Molecular Weight:434.47Molecular Formula:C24,/sub>H23,/sub>FN<sub.4< sub=””>O3</sub.4<>Solubility:Soluble in DMSO (up to 33 mg/ml) or in Ethanol (up to 1.7 mg/ml)Physical Properties:Off-white solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 month.Shipping Code:RT -
PJ-34 HCl | PARP1/2 inhibitor
From $56.00CAS:344458-15-7Catalog Number:10-2395Activity:PARP1,2 inhibitorChemical Name:N-(6-Oxo-5,6-dihydrophenanthridin-2-yl)-(N,N-dimethylamino)acetamide hydrochlorideMolecular Weight:331.81Molecular Formula:C17H17N3O2Solubility:Soluble in DMSO (up to 30 mg/ml) or in Water (up to 20 mg/ml).Physical Properties:Yellow solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:RT (des.)Stability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20° for up to 3 months.Shipping Code:RT -
Rucaparib phosphate | PARP1 inhibitor
From $70.00CAS:459868-92-9Catalog Number:10-3321Activity:PARP1 inhibitorChemical Name:8-Fluoro-1,3,4,5-tetrahydro-2-[4-[(methylamino)methyl]phenyl]-6H-pyrrolo[4,3,2-ef][2]benzazepin-6-onAlternate Name:AG-14699; PF01367338Molecular Weight:421.36Molecular Formula:C19H18FN3O • H3PO4Solubility:Soluble in DMSO (up to 25 mg/ml).Physical Properties:Yellow solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.Shipping Code:RT -
UPF-1069 | PARP-2 inhibitor
From $55.00CAS:1048371-03-4Catalog Number:10-3779Activity:PPAR-2 inhibitorChemical Name:5-(2-Oxo-3-phenylethoxy)-1(2H)-isoquinolinoneMolecular Weight:279.29Molecular Formula:C17H13NO3Solubility:Soluble in DMSO (up to 40 mg/ml).Physical Properties:Off-white solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.Shipping Code:RT -
Veliparib 2HCl | PARP 1/2 inhibitor
From $50.00CAS:912445-05-7Catalog Number:10-2419Activity:PARP 1/2 inhibitorChemical Names:2-[(2R)-2-Methyl-2-pyrrolidinyl]-1H-benzimidazole-7-carboxamide dihydrochlorideAlternate Name:ABT-888Molecular Weight:317.22Molecular Formula:C13H16N4O·2HClSolubility:Soluble in DMSO (30 mg/ml); water (40 mg/ml)Physical Properties:White solidPurity:>98% TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO or water may be stored at -20°C for up to 3 months.Shipping Code:RT
