Highly-Selective Kinase Inhibitor Library
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BML-259 | CDK5/p25 inhibitor
From $60.00CAS:267654-00-2Catalog Number:10-1025Activity:CDK5/p25 inhibitorChemical Name:N-(5-isopropyl-thiazol-2-yl)phenylacetamideMolecular Weight:260.36Molecular Formula:C14H16N2OSSolubility:Soluble in DMSO (up to 25 mg/ml).Physical Properties:white solidPurity:98% by TLCStorage Temperature:RTStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
Chroman 1 | ROCK II inhibitor / Stem cell cytoprotectant
From $45.00CAS:1273579-40-0Catalog Number:10-4912Activity:ROCK II inhibitor / Stem cell cytoprotectantChemical Names:(3S)-N-[2,[2-(Dimethylamino)ethoxy)-4-(1H-pyrazol-4-yl)phenyl]-6-methoxy-3,4-dihydro-2H-chromen-3-carboxamideMolecular Weight:436.51Molecular Formula:C24H28N4O4Solubility:Soluble in DMSO (at least 50 mg/ml)Physical Properties:White solidPurity:99% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.Shipping Code:RT -
Crenolanib | PDGFR and FLT3 inhibitor
From $60.00CAS:670220-88-9Catalog Number:10-4782Activity:PDGFR and FLT3 inhibitorChemical Name:1-[2-[5-[(3-Methyloxetan-3-yl)methoxy]benzimidazole-1-yl]quinoline-8-yl]piperidin-4-amineAlternate Name:CP-868,596Molecular Weight:443.55Molecular Formula:C26H29N5O2Solubility:Soluble in DMSO (up to 15 mg/ml) or in Ethanol (up to 10 mg/ml).Physical Properties:White solidPurity:>97% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 1 month.Shipping Code:RT -
Dabrafenib | B-Raf mutant inhibitor
From $40.00CAS:1195765-45-7Catalog Number:10-1569Activity:B-Raf mutant inhibitorChemical Name:N-[3-[5-(2-amino-4-pyrimidinyl)-2-(1,1-dimethylethyl)-4-thiazolyl]-2-fluorophenyl]-2,6-difluoro-benzenesulfonamideAlternate Names:GSK2118436Molecular Weight:519.56Molecular Formula:C23H20F3N5O2SSolubility:Soluble in DMSO (up to 30 mg/ml with warming), or in Ethanol (up to 1 mg/ml with warming).Physical Properties:Off-white solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.Shipping Code:RT -
Deucravacitinib | Allosteric TYK2 inhibitor
From $100.00CAS:1609392-27-9Catalog Number:10-4756Activity:Allosteric TYK2 inhibitorChemical Names:6-(Cyclopropanecarbonylamino)-4-[2-methoxy-3-(1-methyl-1,2,4-triazol-3-yl)anilino]-N-(trideuteriomethyl)pyridazine-3-carboxamideAlternate Name:BMS-986165Molecular Weight:425.47Molecular Formula:C20H19D3N8O3Solubility:Soluble in DMSO (25 mg/ml with warming); ethanol (20 mg/ml)Physical Properties:White to off-white solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT
