Highly-Selective Kinase Inhibitor Library
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GSK2656157 | PERK inhibitor
From $40.00CAS:1337532-29-2Catalog Number:10-4855Activity:PERK inhibitorChemical Names:1-[5-(4-Amino-7-methylpyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoro-2,3-dihydroindol-1-yl]-2-(6-methylpyridin-2-yl)ethanoneMolecular Weight:416.45Molecular Formula:C23H21FN6OSolubility:Soluble in DMSO (10 mg/ml with warming)Physical Properties:White solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT -
GSK2982772 | RIP1 inhibitor
From $95.00CAS:1622848-92-3Catalog Number:10-4792Activity:RIP1 kinase inhibitorChemical Names:(S)-5-Benzyl-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b]-[1,4]oxazepin-3-yl)-4H-1,2,4-traizole-3-carboxamide; GSK772Molecular Weight:377.40Molecular Formula:C20H19N5O3Solubility:Soluble in DMSO (>25 mg/ml)Physical Properties:Off-white solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT -
GSK8612 | Highly selective TBK1 inhibitor
From $65.00CAS:2361659-62-1Catalog Number:10-4693Activity:Highly selective TBK1 inhibitorChemical Names:4-[[[5-Bromo-2-[[3-methyl-1-(2,2,2-trifluoroethyl)pyrazol-4-yl]amino]pyrimidin-4-yl]amino]methyl]benzenesulfonamideMolecular Weight:520.33Molecular Formula:C17H17BrF3N7O2SSolubility:Soluble in DMSO (20 mg/ml)Physical Properties:Beige solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT -
GW-2580 | cFMS kinase inhibitor
From $72.00CAS:870483-87-7Catalog Number:10-2143Activity:cFMS kinase inhibitorChemical Name:5-(3-Methoxy-4-((4-methoxybenzyl)oxy)benzyl)pyrimidine-2,4-diamineMolecular Weight:366.32Molecular Formula:C20H22N4O3Solubility:Soluble in DMSO (up to 40 mg/ml).Physical Properties:Off-white solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.Shipping Code:RT -
GW-441756 | NGFR kinase inhibitor
From $70.00CAS:504433-23-2Catalog Number:10-1023Activity:NGFR kinase inhibitorChemical Name:1,3-Dihydro-3-[(1-methyl-1H-indol-3-yl)methylene]-2H-pyrrolo[3,2-b]pyridin-2-oneMolecular Weight:275.31Molecular Formula:C17H13N3OSolubility:Soluble in DMSO (up to 5 mg/ml).Physical Properties:Orange solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT
