Inhibitors

  • SKPin C1 | Ubiquitin ligase E3 SCF-Skp2 inhibitor

    CAS:
    432001-69-9
    Catalog Number:
    10-1441
    Activity:
    Ubiquitin ligase E3 SCF-Skp2 inhibitor
    Chemical Names:
    2-[4-Bromo-2-[[4-oxo-3-(3-pyridinyl¬methyl)-2-thioxo-5-thiazolidinylidene]methyl]-phenoxy]acetic acid
    Molecular Weight:
    465.34
    Molecular Formula:
    C18H13BrN2O4S2
    Solubility:
    Soluble in DMSO (15 mg/ml with warming)
    Physical Properties:
    Yellow solid
    Purity:
    98% TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 month.
    Shipping Code:
    RT
    From $70.00
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  • SMI-4a | PIM1 inhibitor

    CAS:
    438190-29-5
    Catalog Number:
    10-1359
    Activity:
    PIM1 inhibitor
    Chemical Name:
    5-(3-Trifluoromethylbenzylidene)thiazolidine
    Molecular Weight:
    273.23
    Molecular Formula:
    C11H6F3NO2S
    Solubility:
    Soluble in DMSO (up to 100 mg/ml) or in Ethanol (up to 40 mg/ml with warming).
    Physical Properties:
    Tan solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 2 months.
    Shipping Code:
    RT
    From $60.00
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  • Taxol | Microtubule stabilizing agent

    CAS:
    33069-62-4
    Catalog Number:
    10-2095
    Activity:
    Microtubule stabilizing agent
    Alternate Names:
    Paclitaxel
    Molecular Weight:
    853.91
    Molecular Formula:
    C47H51NO14
    Solubility:
    Soluble in DMSO (up to 50 mg/ml).
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.
    Shipping Code:
    RT
    From $30.00
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  • Thiostrepton | Antibiotic and FOXM1 inhibitor

    CAS:
    1393-48-2
    Catalog Number:
    10-2108
    Activity:
    Antibiotic and FOXM1 inhibitor
    Chemical Name:
    Fermentation product from Streptomyces azureus
    Molecular Weight:
    1664.91
    Molecular Formula:
    C72H85N19O185
    Solubility:
    Soluble in DMSO (up to 15 mg/ml), or in Chloroform (up to 5 mg/ml).
    Physical Properties:
    Off-white solid
    Purity:
    98% by TLC and HPLC
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 1 week.
    Shipping Code:
    RT
    From $85.00
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  • Tomentosin | Inhibits NFkB activation

    CAS:
    33649-15-9
    Catalog Number:
    10-3538
    Activity:
    Inhibits NFkB activation
    Alternate Names:
    Xanthalongin
    Chemical Name:
    Sesquiterpenoid isolated from Inula viscosa
    Molecular Weight:
    248.32
    Molecular Formula:
    C15H20O3
    Solubility:
    Soluble in DMSO (50 mg/ml)
    Physical Properties:
    Yellow oil
    Purity:
    97% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 month.
    Shipping Code:
    RT
    From $75.00
    View Product This product has multiple variants. The options may be chosen on the product page
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