RGN6024 | Tubulin destabilizer
Available Options
| Size: | Price | Quantity | |
|---|---|---|---|
| 5 mg | $100.00 | ||
| 25 mg | $350.00 |
RGN6024 (3055038-20-2) is an orally bioavailable and brain-penetrant tubulin destabilizer. It inhibits microtubule polymerization by binding to the colchicine binding site of ß-tubulin. Active in glioblastoma cell lines with nanomolar potency. RGN6024 was active in vivo in temozolomide-resistant LN-18 and BT142 glioblastoma xenograft models
References/Citations:
- Patron et al. (2025), RGN6024 Is a Brain-Penetrant, Small-Molecule Tubulin Destabilizer for the Treatment for Glioblastoma; Mol. Cancer Ther. 24 1129
Safety Data Sheet:
Product Data Sheet:
Materials provided by Focus Biomolecules are for laboratory research use only and are not intended for human or veterinary applications. Please note that we do not sell to individuals and that all orders placed by non-research organizations will incur a $20 restocking/refund fee
RGN6024 (3055038-20-2) is an orally bioavailable and brain-penetrant tubulin destabilizer. It inhibits microtubule polymerization by binding to the colchicine binding site of ß-tubulin. Active in glioblastoma cell lines with nanomolar potency. RGN6024 was active in vivo in temozolomide-resistant LN-18 and BT142 glioblastoma xenograft models
References/Citations:
- Patron et al. (2025), RGN6024 Is a Brain-Penetrant, Small-Molecule Tubulin Destabilizer for the Treatment for Glioblastoma; Mol. Cancer Ther. 24 1129
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