Bromocriptine mesylate | Dopamine D2/D3 agonist

CAS:
22260-51-1
Catalog Number:
10-1096
Activity:
Dopamine D2/D3 agonist
Chemical Name:
(+)-2-Bromo-12′-hydroxy-2′-(1-methylethyl)-5′-(2-methylpropyl)-ergotaman-3′,6′,18-trione methanesulfonate
Molecular Weight:
750.72
Molecular Formula:
C32H40BrN5O5·CH3SO3H
Solubility:
Soluble in DMSO (up to 50 mg/ml) or in Ethanol (up to 6 mg/ml).
Physical Properties:
White solid
Purity:
>98% by TLC
NMR (Conforms)
Storage Temperature:
RT
Stability:
Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months
Shipping Code:
RT

Available Options

size :PriceQuantity 
100mg$65.00
500mg$260.00

Bromocriptine mesylate (22260-51-1) is a dopamine D2 receptor agonist.1,2 Inhibits prolactin production.3 Decreases cocaine self-administration in the rat.4 Active in vivo.

References/Citations:

1) Nilsson and Hokfelt (1978), Effect of the dopamine agonist bromocriptine on blood pressure, catecholamines and renin activity in acromegalics at rest, following exercise, and during insulin induced hypoglycemia; Acta Endocrinol., Supp. 216 83
2) Seeman and Van Tol (1994), Dopamine receptor pharmacology;
Trends Pharmacol. Sci., 15 264
3) Carvalho et al. (2015), Maternal prolactin inhibition causes changes in leptin at 22- and 30-day old pups;
Horm. Metab. Res., 47 528
4) Hubner and Koob (1990), Bromocriptine produces decreases in cocaine self-administration in the rat;
Neuropsychopharmacol., 3 101

CAS:
22260-51-1
Catalog Number:
10-1096
Activity:
Dopamine D2/D3 agonist
Chemical Name:
(+)-2-Bromo-12′-hydroxy-2′-(1-methylethyl)-5′-(2-methylpropyl)-ergotaman-3′,6′,18-trione methanesulfonate
Molecular Weight:
750.72
Molecular Formula:
C32H40BrN5O5·CH3SO3H
Solubility:
Soluble in DMSO (up to 50 mg/ml) or in Ethanol (up to 6 mg/ml).
Physical Properties:
White solid
Purity:
>98% by TLC
NMR (Conforms)
Storage Temperature:
RT
Stability:
Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months
Shipping Code:
RT

Safety Data Sheet:

N/A

Product Data Sheet:

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