Bromodomains
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GSK6853 | BRPF1 inhibitor
From $65.00CAS:1910124-24-1Catalog Number:10-4016Activity:BRPF1 inhibitorChemical Names:N-[1,3-Dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamideMolecular Weight:409.49Molecular Formula:C22H27N5O3Solubility:Soluble in DMSO (25 mg/ml); ethanol (25 mg/ml)Physical Properties:White solidPurity:98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.Shipping Code:RT -
I-BET762 | BET Bromodomain inhibitor / Suppresses Myc transcription
From $80.00CAS:1260907-17-2Catalog Number:10-4122Activity:BET Bromodomain inhibitor / Supresses Myc transcriptionChemical Name:(4S)- 6-(4-Chlorophenyl)-N-ethyl-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine-4-acetamideAlternate Names:GSK525762Molecular Weight:423.90Molecular Formula:C22H22ClN5O2Solubility:Soluble in DMSO (up to at least 25 mg/ml) or in Ethanol (up to at least 25 mg/ml)Physical Properties:Tan solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.Shipping Code:RT -
JQ1 (+) | BET Bromodomain inhibitor
From $100.00CAS:1268524-70-4Catalog Number:10-1584Activity:BET Bromodomain inhibitorChemical Name:(6S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid 1,1-dimethylethyl esterMolecular Weight:456.99Molecular Formula:C23H25ClN4O2SSolubility:Soluble in DMSO (up to 60 mg/ml) or in Ethanol (up to 46 mg/ml).Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 2 months.Shipping Code:RT -
JQ1 | Bromodomain inhibitor
From $65.00CAS:1268524-69-1Catalog Number:10-1361Activity:Bromodomain inhibitorChemical Name:(6R,S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid 1,1-dimethylethyl esterMolecular Weight:457Molecular Formula:C23H25ClN4O2SSolubility:Soluble in DMSO (up to 9 mg/ml) or in Ethanol (up to 9 mg/ml).Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 2 months.Shipping Code:RT
