Bromodomains
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PFI-3 | Selective Bromodomain family VIII inhibitor
From $59.00CAS:1819363-80-8Catalog Number:10-4034Activity:Selective Bromodomain family VIII inhibitorChemical Names:(2E)-1-(2-Hydroxyphenyl)-3-[(1R,4R)-5-(pyridine-2-yl)-2,5-diazabicyclo{2.2.1]heptan-2-yl]prop-2-en-1-oneMolecular Weight:321.37Molecular Formula:C19H19N3O2Solubility:Soluble in DMSO (>25 mg/ml)Physical Properties:Yellow solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT -
RVX-208 | BET bromodomain inhibitor
From $68.00CAS:1044870-39-4Catalog Number:10-1487Activity:BET bromodomain inhibitorChemical Name:2-[4-(2-hydroxyethoxy)-3,5-dimethylphenyl]-5,7-dimethoxy-4(3H)-quinzolinoneMolecular Weight:370.41Molecular Formula:C20H22N2O5Solubility:Soluble in DMSO (up to 75 mg/ml) or in Ethanol (up to 4 mg/ml).Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°C (des.)Stability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 1 month.Shipping Code:RT -
Volasertib | Potent and selective inhibitor of Polo-like kinase 1
From $80.00CAS:755038-65-4Catalog Number:10-4818Activity:Potent and selective inhibitor of Polo-like kinase 1Chemical Name:N-[4-[4-(Cyclopropylmethyl)piperazin-1-yl]cyclohexyl]-4-[[(7R)-7-ethyl-5-methyl-6-oxo-8-propan-2-yl-7H-pteridin-2-yl]amino]-3-methoxybenzamideAlternate Name:BI 6727Molecular Weight:618.82Molecular Formula:C34H50N8O3Solubility:Soluble in DMSO (up to at least 25 mg/ml).Physical Properties:Off-white solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 1 month.Shipping Code:RT
