PARP

  • 3-Aminobenzamide | PARP inhibitor

    CAS:
    3544-24-9
    Catalog Number:
    10-1239
    Activity:
    PARP inhibitor
    Alternate Names:
    3-AB
    Molecular Weight:
    136.15
    Molecular Formula:
    C7H8N2O
    Solubility:
    Soluble in DMSO (up to 25 mg/ml) or in Ethanol (up to 4 mg/ml).
    Physical Properties:
    White to tan solid
    Purity:
    97% by TLC
    NMR (Conforms)
    Storage Temperature:
    RT
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    $50.00
  • ME-0328 | PARP3 inhibitor

    CAS:
    1445251-22-8
    Catalog Number:
    10-1484
    Activity:
    PARP3 inhibitor
    Chemical Name:
    3,4-Dihydro-4-oxo-3,4-Dihydro-4-oxo-N-[(1S)-1-phenylethyl]-2-quinazolinepropanamide
    Molecular Weight:
    321.38
    Molecular Formula:
    C19H19N3O2
    Solubility:
    Soluble in DMSO (up to 30 mg/ml), or in Ethanol (up to 4 mg/ml with warming).
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    RT
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months.
    Shipping Code:
    RT
    From $70.00
  • Olaparib | PARP1 inhibitor

    CAS:
    763113-22-0
    Catalog Number:
    10-2154
    Activity:
    PARP1 inhibitor
    Chemical Name:
    4-(3-(4-(Cyclopropanecarbonyl)piperazine-1-carbonyl)-4-fluorobenzyl)phthalazine-1(2H)-one
    Alternate Names:
    AZD-2281; KU-59436
    Molecular Weight:
    434.47
    Molecular Formula:
    C24,/sub>H23,/sub>FN<sub.4< sub=””>O3</sub.4<>
    Solubility:
    Soluble in DMSO (up to 33 mg/ml) or in Ethanol (up to 1.7 mg/ml)
    Physical Properties:
    Off-white solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $45.00
  • PJ-34 HCl | PARP1/2 inhibitor

    CAS:
    344458-15-7
    Catalog Number:
    10-2395
    Activity:
    PARP1,2 inhibitor
    Chemical Name:
    N-(6-Oxo-5,6-dihydrophenanthridin-2-yl)-(N,N-dimethylamino)acetamide hydrochloride
    Molecular Weight:
    331.81
    Molecular Formula:
    C17H17N3O2
    Solubility:
    Soluble in DMSO (up to 30 mg/ml) or in Water (up to 20 mg/ml).
    Physical Properties:
    Yellow solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    RT (des.)
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20° for up to 3 months.
    Shipping Code:
    RT
    From $56.00
  • Rucaparib phosphate | PARP1 inhibitor

    CAS:
    459868-92-9
    Catalog Number:
    10-3321
    Activity:
    PARP1 inhibitor
    Chemical Name:
    8-Fluoro-1,3,4,5-tetrahydro-2-[4-[(methylamino)methyl]phenyl]-6H-pyrrolo[4,3,2-ef][2]benzazepin-6-on
    Alternate Name:
    AG-14699; PF01367338
    Molecular Weight:
    421.36
    Molecular Formula:
    C19H18FN3O • H3PO4
    Solubility:
    Soluble in DMSO (up to 25 mg/ml).
    Physical Properties:
    Yellow solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.
    Shipping Code:
    RT
    From $70.00