Highly Selective Inhibitors
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AZD1152-HQPA | Aurora B kinase inhibitor
From $50.00CAS:722544-51-6Catalog Number:10-4804Activity:Aurora B kinase inhibitorChemical Name:3-[[7-[3-[Ethyl(2-hydroxyethyl)amino]propoxy]-4-quinazolinyl]amino-N-(3-fluorophenyl)-1H-pyrazole-5-acetamideAlternate Name:Barasertib-HQPA; AZD2811Molecular Weight:507.56Molecular Formula:C26H30FN7O3Solubility:Soluble in DMSO (up to 15 mg/ml).Physical Properties:Yellow solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 1 month.Shipping Code:RT -
AZD6244 | ERK inhibitor
From $40.00CAS:606143-52-6Catalog Number:10-4509Activity:ERK inhibitorAlternate Names:ARRY-142886, SelumetinibMolecular Weight:457.68Molecular Formula:C17H15BrClFN4O3Solubility:Soluble in DMSO (up to 50 mg/ml) or in Ethanol (up to 2 mg/ml)Physical Properties:White solidPurity:99% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 2 months.Shipping Code:RT -
AZD8055 | mTOR kinase inhibitor
From $45.00CAS:1009298-09-2Catalog Number:10-4816Activity:mTOR kinase inhibitorChemical Name:(5-(2,4-bis((3S)-3-methylmorpholin-4-yl)pyrido(2,3-d)pyrimidin-7-yl)-2-methoxyphenyl)methanolMolecular Weight:465.54Molecular Formula:C25H31N5O4Solubility:Soluble in DMSO (up to 30 mg/ml)Physical Properties:Yellow solidPurity:99% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.Shipping Code:RT -
Binimetinib | MEK1/2 inhibitor
From $39.00CAS:606143-89-9Catalog Number:10-4789Activity:MEK1/2 inhibitorChemical Name:6-(4-Bromo-2-fluoroanilino)-7-fluoro-N-(2-hydroxyethoxy)-3-methylbenzimidazole-5-carboxamideAlternate Names:ARRY-162; MEK162Molecular Weight:441.23Molecular Formula:C17H15BrF2N4O3Solubility:Soluble in DMSO (up to at least 25 mg/ml)Physical Properties:White solidPurity:99% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
Duvelisib | PI3Kdelta/gamma inhibitor
From $65.00CAS:1201438-56-3Catalog Number:10-4788Activity:PI3Kδ/γ inhibitor/Cancer immunotherapy enhancerChemical Name:8-Chloro-2-phenyl-3-[(1S)-1-(7H-purin-6-ylamino)ethyl]isoquinolin-1-oneAlternative Name:IPI-145Molecular Weight:416.87Molecular Formula:C22H17ClN6OSolubility:Soluble in DMSO (up to at least 25 mg/ml)Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT
