Antagonists

  • BD1047 dihydrobromide | Selective sigma-1 antagonist

    CAS:
    138356-21-5
    Catalog Number:
    10-4210
    Activity:
    Selective sigma-1 antagonist
    Chemical Name:
    N-[2-(3,4Dichlorophenyl)ethyl]-N-methyl-2-(dimethylamino)ethylamine dihydrobromide
    Molecular Weight:
    437.04
    Molecular Formula:
    C13H20Cl2N2 • 2HBr
    Solubility:
    Soluble in DMSO (up to 20 mg/ml) or in Water (up to 20 mg/ml)
    Physical Properties:
    Off-white solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $50.00
  • BD1063 dihydrochloride | Selective sigma-1 antagonist

    CAS:
    206996-13-6
    Catalog Number:
    10-4211
    Activity:
    Selective sigma-1 antagonist
    Chemical Name:
    1-[2-(3,4-Dichlorophenyl)ethyl]-4-methylpiperazine dihydrochloride
    Molecular Weight:
    346.13
    Molecular Formula:
    C13H18Cl2N2 • 2HCl
    Solubility:
    Soluble in Water (up to at least 25 mg/ml)
    Physical Properties:
    Off-white solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in distilled water may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $50.00
  • NE-100 | Selective sigma-1 antagonist

    CAS:
    149409-57-4
    Catalog Number:
    10-4200
    Activity:
    Selective sigma-1 antagonist
    Chemical Name:
    4-Methoxy-3-(2-phenylethoxy)-N,N,dipropylbenzeneethanamine hydrochloride
    Molecular Weight:
    391.97
    Molecular Formula:
    C23H33NO2 • HCl
    Solubility:
    Soluble in DMSO (up to at least 25 mg/ml) or in Water (up to 10 mg/ml)
    Physical Properties:
    White solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $70.00
  • S1RA | Selective sigma-1 antagonist

    CAS:
    1265917-14-3
    Catalog Number:
    10-4201
    Activity:
    Selective Sigma1 antagonist
    Chemical Name:
    4-{2-[5-Methyl-1-(napthalen-2-yl)-1H-pyrazol-3-yloxy]ethyl}morpholine hydrochloride
    Alternate Names:
    E-52862 HCl
    Molecular Weight:
    373.88
    Molecular Formula:
    C20H23N3O2 • HCl
    Solubility:
    Soluble in DMSO (up to at least 25 mg/ml)
    Physical Properties:
    Off-white solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C (des.)
    Stability:
    Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $85.00

EXPLORE OTHER Sigma Receptor