Polycomb Repressive Complex Library
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DZNep HCl | Methyltransferase inhibitor
From $142.00CAS:120964-45-6Catalog Number:10-1524Activity:Methyl transferase inhibitorChemical Name:(1S,2R,5R)-5-(4-Aminoimidazo[4,5-c]pyridine-1-yl)-3-(hydroxymethyl)-cyclopent-3-ene-1,2-diol hydrochlorideAlternate Names:3-Deazaneplanocin A HCl; NSC 617989Molecular Weight:298.73Molecular Formula:C12H14N4O3 ·HClSolubility:Soluble in Water (up to 40 mg/ml)Physical Properties:Beige solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in water may be stored at -20°C for up to 1 month.Shipping Code:RT -
EED-226 | PRC2 methyltransferase inhibitor
From $85.00CAS:2083627-02-3Catalog Number:10-4021Activity:PRC2 methyltransferase inhibitorChemical Name:N-(Furan-2-ylmethyl)-8-(4-methylsulfonylphenyl)-[1,2,4]triazolol[4,3-c)pyrimidine-5-amineMolecular Weight:369.40Molecular Formula:C17H15N5O3SSolubility:Soluble in DMSO (up to 25 mg/ml).Physical Properties:Off-white solidPurity:98% by HPLCNMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 1 month.Shipping Code:RT -
PRT4165 | E3 ubiquitin ligase inhibitor
From $65.00CAS:31083-55-3Catalog Number:10-1478Activity:E3 ubiquitin ligase inhibitorChemical Name:2-(3-Pyridinylmethylene)-1H-indene-1,3(2H)-dioneMolecular Weight:235.24Molecular Formula:C15H9NO2Solubility:Soluble in DMSO (up to 25 mg/ml) or in Ethanol (up to 6 mg/ml with warming).Physical Properties:Yellow solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.Shipping Code:RT -
PTC-209 | BMI-1 inhibitor
From $60.00CAS:315704-66-6Catalog Number:10-4022Activity:BMI-1 inhibitorChemical Names:N-(2,6-Dibromo-4-methoxyphenyl)-4-(2-methylimidazol[1,2-a]pyrimidin-3-yl)-2-thiazolamineMolecular Weight:495.19Molecular Formula:C17H13Br2N5OSSolubility:Soluble in DMSO (>25 mg/ml)Physical Properties:Yellow solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
Tazemetostat | EZH2 inhibitor
From $55.00CAS:1403254-99-8Catalog Number:10-4032Activity:EZH2 inhibitorChemical Name:N-((4,6-Dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-5-(ethyl(tetrahydro-2H-pyran-4-yl)amino)-4-methyl-4’-(morpholinomethyl)-[1,1’-biphenyl]-3-carboxamideAlternate Name:EPZ-6438Molecular Weight:572.75Molecular Formula:C34H44N4O4Solubility:Soluble in DMSO (up to at least 25 mg/ml).Physical Properties:Off-white solidPurity:98%NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 1 month.Shipping Code:RT
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