Pain
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S1RA | Selective sigma-1 antagonist
From $85.00CAS:1265917-14-3Catalog Number:10-4201Activity:Selective Sigma1 antagonistChemical Name:4-{2-[5-Methyl-1-(napthalen-2-yl)-1H-pyrazol-3-yloxy]ethyl}morpholine hydrochlorideAlternate Names:E-52862 HClMolecular Weight:373.88Molecular Formula:C20H23N3O2 • HClSolubility:Soluble in DMSO (up to at least 25 mg/ml)Physical Properties:Off-white solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°C (des.)Stability:Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
SB-705498 | TRPV1 blocker
From $65.00CAS:501951-42-4Catalog Number:10-3985Activity:TRPV1 blockerChemical Names:1-(2-Bromophenyl)-3-[(3R)-1-[5-(trifluoromethyl)pyridine-2-yl]pyrrolidine-3-yl]ureaMolecular Weight:429.24Molecular Formula:C17H16BrF3N4OSolubility:Soluble in DMSO (>25 mg/ml)Physical Properties:White solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
SC-51089 | Prostaglandin E2 (EP1) antagonist
From $55.00CAS:146033-02-5Catalog Number:10-1135Activity:PGE2 (EP1 receptor) antagonistChemical Names:8-Chlorodibenz(Z)[b,f]oxazepine-10(11H)-carboxylic acid 2-[1-oxo-3-(4-pyridinyl)propyl]hydrazide hydrochlorideMolecular Weight:459.34Molecular Formula:C22H19ClN4O3·HClSolubility:Soluble in DMSO (25 mg/ml) or water (25 mg/mL)Physical Properties:White solidPurity:98% TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 3 months.Shipping Code:RT -
Serodolin | ß-Arrestin-biased 5-HT7 antagonist
From $80.00CAS:1814929-81-1Catalog Number:10-4086Activity:ß-Arrestin-biased 5-HT7 antagonistChemical Names:1-(5-(4-(4-Fluorophenyl)piperazin-1-yl)pentyl)-1H-benzo[d]imidazole-2(3H)-oneMolecular Weight:382.47Molecular Formula:C22H27FN4OSolubility:Soluble in DMSO (at least 50 mg/ml)Physical Properties:Off-white solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
SR-144528 | Cannabinoid CB2 antagonist
From $100.00CAS:192703-06-3Catalog Number:10-1164Activity:Cannabinoid CB2 antagonistChemical Name:5-(4-Chloro-3-methylphenyl)-1-[(4-methylphenyl)methyl]-N-[(1S,2S,4R)-1,3,3-trimethylbicyclo[2.2.1]hept-2-yl]-1H-pyrazole-3-carboxamideMolecular Weight:476.07Molecular Formula:C29H34ClN3OSolubility:Soluble in DMSO (up to 20 mg/ml, with warming).Physical Properties:Off-white solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT
