Pain

  • SC-51089 | Prostaglandin E2 (EP1) antagonist

    CAS:
    146033-02-5
    Catalog Number:
    10-1135
    Activity:
    PGE2 (EP1 receptor) antagonist
    Chemical Names:
    8-Chlorodibenz(Z)[b,f]oxazepine-10(11H)-carboxylic acid 2-[1-oxo-3-(4-pyridinyl)propyl]hydrazide hydrochloride
    Molecular Weight:
    459.34
    Molecular Formula:
    C22H19ClN4O3·HCl
    Solubility:
    Soluble in DMSO (25 mg/ml) or water (25 mg/mL)
    Physical Properties:
    White solid
    Purity:
    98% TLC
    NMR (Conforms)
    Storage Temperature:
    RT
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $55.00
  • Serodolin | ß-Arrestin-biased 5-HT7 antagonist

    CAS:
    1814929-81-1
    Catalog Number:
    10-4086
    Activity:
    ß-Arrestin-biased 5-HT7 antagonist
    Chemical Names:
    1-(5-(4-(4-Fluorophenyl)piperazin-1-yl)pentyl)-1H-benzo[d]imidazole-2(3H)-one
    Molecular Weight:
    382.47
    Molecular Formula:
    C22H27FN4O
    Solubility:
    Soluble in DMSO (at least 50 mg/ml)
    Physical Properties:
    Off-white solid
    Purity:
    >98% HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $80.00
  • SR-144528 | Cannabinoid CB2 antagonist

    CAS:
    192703-06-3
    Catalog Number:
    10-1164
    Activity:
    Cannabinoid CB2 antagonist
    Chemical Name:
    5-(4-Chloro-3-methylphenyl)-1-[(4-methylphenyl)methyl]-N-[(1S,2S,4R)-1,3,3-trimethylbicyclo[2.2.1]hept-2-yl]-1H-pyrazole-3-carboxamide
    Molecular Weight:
    476.07
    Molecular Formula:
    C29H34ClN3O
    Solubility:
    Soluble in DMSO (up to 20 mg/ml, with warming).
    Physical Properties:
    Off-white solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $100.00
  • SR-9009 | RevErb alpha/beta agonist

    CAS:
    1379686-30-2
    Catalog Number:
    10-1511
    Activity:
    RevErbα/β agonist
    Chemical Name:
    Ethyl 3-(((4-chlorobenzyl)((5-nitrophen-2-yl)methyl)amino)methyl)pyrrolidine-1-carboxylate hydrochloride
    Molecular Weight:
    474.4
    Molecular Formula:
    C20H24CLN3O4S HCl
    Solubility:
    Soluble in DMSO (greater than 25 mg/ml) or in Ethanol (up to 20 mg/ml).
    Physical Properties:
    Tan solid
    Purity:
    98% by TLC
    Storage Temperature:
    -20°
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 1 month.
    Shipping Code:
    RT
    From $70.00
  • ST034307 | Adenylate cyclase 1 inhibitor/analgesic activity

    CAS:
    133406-29-8
    Catalog Number:
    10-1620
    Activity:
    Adenylate cyclase 1 inhibitor/analgesic activity
    Chemical Name:
    6-Chloro-2-(trichloromethyl)-4H-1-benzopyran-4-one
    Molecular Weight:
    297.95
    Molecular Formula:
    C10H4Cl4O2
    Solubility:
    Soluble in DMSO (up to 30 mg/ml) or in Ethanol (up to 6 mg/ml)
    Physical Properties:
    Yellow solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    RT
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $65.00
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