Lipid Receptor Agonists & Antagonists

  • LY-171883 | Cys LT1 antagonist

    CAS:
    88107-10-2
    Catalog Number:
    10-1052
    Activity:
    Cys LT1 antagonist
    Chemical Name:
    1-[2-Hydroxy-3-propyl-4-[4-1H-tetrazol-5-yl)butoxy]phenyl]ethanone
    Molecular Weight:
    318.37
    Molecular Formula:
    C16H22N4O3
    Solubility:
    Soluble in DMSO (up to 30 mg/ml) or in Ethanol (up to 15 mg/ml),
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C (des.)
    Stability:
    Stable for 2 years as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months
    Shipping Code:
    RT
    From $60.00
  • MK-571 | Cys LT1 antagonist

    CAS:
    115104-28-4
    Catalog Number:
    10-1039
    Activity:
    Cys LT1 antagonist
    Alternate Names:
    L-660711
    Chemical Name:
    5-(3-(2-(7-Chloroquinolin-2-yl)ethenyl)phenyl)-8-dimethylcarbamyl-4,6-dithiaoctanoic acid
    Molecular Weight:
    515.09
    Molecular Formula:
    C26H27ClN2O3S2
    Solubility:
    Soluble in DMSO (up to 50 mg/ml).
    Physical Properties:
    Yellow solid
    Purity:
    95% by TLC
    NMR (Conforms)
    Storage Temperature:
    RT
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.
    Shipping Code:
    RT
    From $60.00
  • Montelukast sodium | Leukotriene antagonist and GPR17 antagonist

    CAS:
    151767-02-1
    Catalog Number:
    10-2597
    Activity:
    Leukotriene antagonist and GRP17 antagonist
    Chemical Name:
    2-[1-[[(1R)-1-[3-[(E)-2-(7-Chloroquinolin-2-yl)ethenyl]phenyl]-3-[2-(2-hydroxypropan-2-yl)phenyl]propyl]sulfanylmethyl]cyclopropyl]acetate, sodium salt
    Alternate Names:
    MK-0476
    Molecular Weight:
    608.17
    Molecular Formula:
    C35H35ClNO3S
    Solubility:
    Soluble in DMSO (up to 60 mg/ml), in Water (up to 30 mg/ml) , or in Ethanol (up to 60 mg/ml)
    Physical Properties:
    Solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO, distilled water, or ethanol may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $60.00
  • N-Arachidonoyldopamine | Endogenous TRPV1 activator

    CAS:
    199875-69-9
    Catalog Number:
    10-1479
    Activity:
    Endogenous TRPV1 activator
    Chemical Name:
    N-(5Z,8Z,11Z,14Z-eicosatetraenoyl)dopamine
    Alternate Name:
    NADA; AA-DA
    Molecular Weight:
    439.63
    Molecular Formula:
    C28H41NO3
    Solubility:
    Soluble in DMSO (up to 50 mg/ml).
    Physical Properties:
    Pale yellow viscous oil
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -80° (des.)
    Stability:
    Stable for 2 years from date of purchase as supplied. Subject to air oxidation Solutions in DMSO may be stored at -80° under an inert atmosphere for up to 1 month.
    Shipping Code:
    Blue Ice
    From $46.00
  • NA-Gly | GPR18 agonist

    CAS:
    179113-91-8
    Catalog Number:
    10-1200
    Activity:
    GPR18 agonist
    Alternate Names:
    N-Arachidonylglycine
    Chemical Name:
    N-(5Z,8Z,11Z,14Z-eicosatetraenoyl)glycine
    Molecular Weight:
    361.53
    Molecular Formula:
    C22H35NO3
    Solubility:
    Soluble in DMSO (up to 50 mg/ml).
    Physical Properties:
    Beige waxy solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Product is subject to oxidation. Solutions in degassed DMSO may be stored at -20°C for up to 1 month.
    Shipping Code:
    Blue Ice
    From $60.00
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