Histone Demethylation
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DMOG | Inhibits prolyl hydroxylase domain-containing proteins
From $60.00CAS:89464-63-1Catalog Number:10-2371Activity:Inhibits prolyl hydroxylase domain-containing proteinsAlternate Names:DimethyloxalylglycineChemical Name:N-(2-Methoxy-2-oxoacetyl)glycine methyl esterMolecular Weight:175.14Molecular Formula:C6H9NO5Solubility:Soluble in DMSO (up to 25 mg/ml) or in Ethanol (up to 25 mg/ml).Physical Properties:Off-white solidPurity:99% by TLC
NMR (Conforms)Storage Temperature:-20°C
Protect from lightStability:Stable for 2 years from date of purchase as supplied. Solutions are not stable. Solutions must be made fresh and used within 1 working day.Shipping Code:RT -
GSK-J1 | JMJ H3K27 Demethylase inhibitor (Non-cell permeable)
From $75.00CAS:1373422-53-7Catalog Number:10-1393Activity:JMJ H3K27 Demethylase inhibitor (Non-cell permeable)Chemical Name:N-[2-(2-Pyridinyl)-6-(1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl)-4-pyrimidinyl]-β-alanineMolecular Weight:389.46Molecular Formula:C22H23N5O2Solubility:Soluble in DMSO (up to 20 mg/ml).Physical Properties:Pale yellow solidPurity:99% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.Shipping Code:RT -
GSK-J4 | JMJ H3K27 Demethylase inhibitor (Cell Permeable)
From $50.00CAS:1373423-53-0Catalog Number:10-1394Activity:JMJ H3K27 Demethylase inhibitor (Cell Permeable)Chemical Name:N-[2-(2-Pyridinyl)-6-(1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl)-4-pyrimidinyl]-β-alanine ethyl esterMolecular Weight:417.48Molecular Formula:C24H27N5O2Solubility:Soluble in DMSO (up to 40 mg/ml) or in Ethanol (up to 40 mg/ml).Physical Properties:Yellow waxy solidPurity:99% by TLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months.Shipping Code:RT -
GSK2879552 | Potent and selective LSD1 inhibitor
From $80.00CAS:1401966-69-5Catalog Number:10-4020Activity:Potent and selective LSD1 inhibitorChemical Name:4-[[4-[[[(1R,2S)-2-Phenylcyclopropyl]amino]methyl]-1-piperidinyl]methyl]benzoic acid dihydrochlorideMolecular Weight:437.40Molecular Formula:C23H28N2O2 • HClSolubility:Soluble in DMSO (up to 25 mg/ml) or in Water (up to at least 25 mg/ml)Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 3 months.Shipping Code:RT
