E3 Ubiquitin ligase
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Lenalidomide | Immunomodulator
From $75.00CAS:191732-72-6Catalog Number:10-2148Activity:ImmunomodulatorChemical Name:(R,S)-3-(4-Amino-1-oxo-3H-isoindol-2-yl)piperidine-2,6-dioneMolecular Weight:259.26Molecular Formula:C13H13N3O3Solubility:Soluble in DMSO (up to 30 mg/ml)Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
NAcM-OPT | NEDD8 ligation inhibitor
From $55.00CAS:2089293-61-6Catalog Number:10-1636Activity:NEDD8 ligation inhibitorChemical Name:1-Benzyl-1-(1-butylpiperidin-4-yl)-3-(3,4-dichlorophenyl)ureaMolecular Weight:434.40Molecular Formula:C23H29Cl2N3OSolubility:Soluble in DMSO (up to 30 mg/ml) or in Ethanol (up to 20 mg/ml)Physical Properties:White solidPurity:98% by HPLC/TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year as from date of purchase supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.Shipping Code:RT -
Pomalidomide | Cereblon ubiquitination inhibitor
From $50.00CAS:19171-19-8Catalog Number:10-2768Activity:Cereblon ubiquination inhibitorChemical Name:1,3-Dioxo-2-(2,6-dioxopiperidin-3-yl)-4-aminoisoindoline; 3-amino-N-(2,6-dioxo-3-piperidyl)phthalamideMolecular Weight:273.24Molecular Formula:C13H11N3O4Solubility:Soluble in DMSO (up to 50 mg/ml).Physical Properties:Yellow solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 1 month.Shipping Code:RT -
PRT4165 | Bmi1/Ring1A inhibitor
From $65.00CAS:31083-55-3Catalog Number:10-1478Activity:Bmi1/Ring1A inhibitorChemical Name:2-(3-Pyridinylmethylene)-1H-indene-1,3(2H)-dioneMolecular Weight:235.24Molecular Formula:C15H9NO2Solubility:Soluble in DMSO (up to 25 mg/ml) or in Ethanol (up to 6 mg/ml with warming).Physical Properties:Yellow solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.Shipping Code:RT -
SKPin C1 | Ubiquitin ligase E3 SCF-Skp2 inhibitor
From $70.00CAS:432001-69-9Catalog Number:10-1441Activity:Ubiquitin ligase E3 SCF-Skp2 inhibitorChemical Names:2-[4-Bromo-2-[[4-oxo-3-(3-pyridinyl¬methyl)-2-thioxo-5-thiazolidinylidene]methyl]-phenoxy]acetic acidMolecular Weight:465.34Molecular Formula:C18H13BrN2O4S2Solubility:Soluble in DMSO (15 mg/ml with warming)Physical Properties:Yellow solidPurity:98% TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 month.Shipping Code:RT
