Protease inhibitors
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GRL-0496 | SARS-CoV 3CLpro inhibitor
From $60.00CAS:1087243-14-8Catalog Number:10-4960Activity:SARS-CoV 3CLpro inhibitorChemical Name:1H-Indole-4-carboxylic acid, 5-chloro-3-pyridinyl esterMolecular Weight:272.69Molecular Formula:C14H9ClN2O2Solubility:Soluble in DMSO (>30 mg/mL) and ethanol (>25 mg/mL)Physical Properties:White solidPurity:>98% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months.Shipping Code:RT -
GRL-0617 | Potent SARS-CoV PLpro inhibitor
From $75.00CAS:1093070-16-6Catalog Number:10-4965Activity:Potent SARS-CoV PLpro inhibitorChemical Name:5-Amino-2-methyl-N-(1R-naphthalen-1-yl-ethyl)benzamideMolecular Weight:304.39Molecular Formula:C20H20N2OSolubility:Soluble in DMSO (>30 mg/mL) and ethanol (15 mg/mL)Physical Properties:Beige solidPurity:99% by HPLC
NMR (Conforms)Storage Temperature:-20° (des.)Stability:Stable for 1 year as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months.Shipping Code:RT -
GRL-0667 | Noncovalent inhibitor of SARS-CoV PLpro
From $95.00CAS:1234195-91-5Catalog Number:10-4963Activity:Noncovalent SARS-CoV Plpro inhibitorChemical Names:1-[(R)-1-(1-Naphthyl)ethyl)]-4-[3,4-(methylenedioxy)benzylamino]carbonylpiperidineMolecular Weight:416.52Molecular Formula:C26H28N2O3Solubility:Soluble in DMSO (>25 mg/ml) or ethanol (15 mg/ml)Physical Properties:Off-white solidPurity:98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 month.Shipping Code:RT -
Nelfinavir mesylate | HIV protease inhibitor / Anticancer activity
From $60.00CAS:159989-65-8Catalog Number:10-3050Activity:HIV protease inhibtior / Anticancer activityChemical Name:(3S,4aS,8aS)-N-(1,1-Dimethylethyl)decahydro-2-[(2R,3R)-2-hydroxy-3-[(3-hydroxy-2-methylbenzoyl)amino]-4-(phenylthio)butyl]-3-isoquinolinecarboxamide methanesulfonateAlternate Name:AG-1343Molecular Weight:663.88Molecular Formula:C32H45N3O4S • CH3SO3HSolubility:Soluble in DMSO (up to 70 mg/ml).Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°Stability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months.Shipping Code:RT -
Ritonavir | HIV1/2 protease inhibitor
From $40.00CAS:155213-67-5Catalog Number:10-4484Activity:HIV 1/2 protease inhibitorChemical Name:1,3-Thiazol-5-ylmethyl N-[(2S,3S,5S)-3-hydroxy-5-[[(2S)-3-methyl-2-[[methyl-2-[(2-propan-2-yl-1,3-thiazol-4-yl)methyl]carbamoyl]amino]butanoyl]amino]-1,6-diphenylhexan-2-yl]carbamateMolecular Weight:720.95Molecular Formula:C37H48N5O5S2Solubility:Soluble in DMSO (up to 12 mg/ml with warming) or in Ethanol (up to 5 mg/ml).Physical Properties:White solidPurity:98% by HPLCStorage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 2 months.Shipping Code:RT
