Epigenetics
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C-DIM 8 | Nur77 Antagonist
From $40.00CAS:151358-47-3Catalog Number:10-5157Activity:Nur77 antagonistChemical Names:1,1-Bis(3’-indolyl)-1-(p-hydroxyphenyl)methaneAlternate Name:DIM-C-pPhOHMolecular Weight:338.41Molecular Formula:C23H18N2OSolubility:Soluble in DMSO (35 mg/ml); ethanol (35 mg/ml)Physical Properties:Pink solidPurity:>98% TLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.Shipping Code:RT -
CI-994 | HDAC Inhibitor
From $38.00CAS:112522-64-2Catalog Number:10-2125Activity:HDAC inhibitorChemical Name:4-(Acetylamino)-N-(2-aminophenyl)benzamideAlternate Names:Tacedinaline; PD-123654; N-acetyl-dinaline; GOE-5549Molecular Weight:269.30Molecular Formula:C15H15N3O2Solubility:Soluble in DMSO (up to 25 mg/ml)Physical Properties:Off-white solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT -
CPI-455 | Lysine demethylase KDM5 inhibitor
From $90.00CAS:1628208-23-0Catalog Number:10-4035Activity:Lysine demethylase KDM5 inhibitorChemical Name:7-Oxo-5-phenyl-6-propan-2-yl-1H-pyrazolo[1,5-a]pyrimidine-3-carbonitrileMolecular Weight:278.32Molecular Formula:C16H14N4OSolubility:Soluble in DMSO (up to at least 25 mg/ml)Physical Properties:Off-white solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
CUDC-101 | Dual HDAC and EGFR inhibitor
From $70.00CAS:1012054-59-9Catalog Number:10-2491Activity:Dual HDAC and EGFR inhibitorChemical Name:7-((4-((3-Ethynylphenyl)amino)-7-methoxyquinazolin-6-yl)oxy)-N-hydroxyheptanamideMolecular Weight:434.49Molecular Formula:C24H26N4O4Solubility:Soluble in DMSO (up to 25 mg/ml)Physical Properties:White or off-white solidPurity:99% by HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT
EXPLORE OTHER Cancer
- ADC warheads
- Angiogenesis
- Autophagy
- Cancer Cell Metabolism
- Cancer Stem Cells
- Cell Cycle
- Cellular Stress
- Chemotherapeutics
- Cytoskeleton
- DNA Damage/Repair
- Drug resistance
- Gene Regulation/Transcription
- Growth factors
- Immuno-oncology
- Kinases
- Metastasis
- Other Cancer
- p53 & Other Tumor Suppressors
- Programmed cell death
- Stem Cells
- Ubiquitin proteasome
- Wnt/ß-Catenin
