Epigenetics
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JQ1 (+) | BET Bromodomain inhibitor
From $100.00CAS:1268524-70-4Catalog Number:10-1584Activity:BET Bromodomain inhibitorChemical Name:(6S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid 1,1-dimethylethyl esterMolecular Weight:456.99Molecular Formula:C23H25ClN4O2SSolubility:Soluble in DMSO (up to 60 mg/ml) or in Ethanol (up to 46 mg/ml).Physical Properties:White solidPurity:98% by HPLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 2 months.Shipping Code:RT -
JQ1 | Bromodomain inhibitor
From $65.00CAS:1268524-69-1Catalog Number:10-1361Activity:Bromodomain inhibitorChemical Name:(6R,S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid 1,1-dimethylethyl esterMolecular Weight:457Molecular Formula:C23H25ClN4O2SSolubility:Soluble in DMSO (up to 9 mg/ml) or in Ethanol (up to 9 mg/ml).Physical Properties:White solidPurity:98% by TLC
NMR (Conforms)Storage Temperature:RTStability:Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 2 months.Shipping Code:RT -
LD2 | PRMT9 inhibitor
From $60.00CAS:1134334-55-6Catalog Number:10-4872Activity:PRMT9 inhibitorChemical Names:4-Chloro-8-methoxy-5-methyl-5H-pyrimido[5,4-b]indoleMolecular Weight:247.68Molecular Formula:C12H10ClN3OSolubility:Soluble in DMSO (at least 40 mg/ml)Physical Properties:Pale yellow solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.Shipping Code:RT -
LMK235 | Selective HDAC4/5 inhibitor
From $60.00CAS:1418033-25-6Catalog Number:10-4024Activity:HDAC4/5 inhibitorChemical Names:N-[6-(Hydroxyamino)-6-oxohexoxy]-3,5-dimethylbenzamideMolecular Weight:294.35Molecular Formula:C15H22N2O4Solubility:Soluble in DMSO (25 mg/ml)Physical Properties:Off-white solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.Shipping Code:RT -
MDL-800 | Allosteric activator of SIRT6
From $85.00CAS:2275619-53-7Catalog Number:10-4415Activity:Allosteric activator of SIRT6Chemical Names:Methyl 2-(N-(5-Bromo-4-fluoro-2-methylphenyl)sulfamoyl)-5-(3,5-dichlorophenylsulfonamido)benzoateMolecular Weight:626.29Molecular Formula:C21H16BrCl2FN2O6S2Solubility:Soluble in DMSO (up to at least 10 mg/ml with warming)Physical Properties:White solidPurity:>98% HPLC
NMR (Conforms)Storage Temperature:-20°CStability:Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.Shipping Code:RT
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