Kinases

  • BI-D1870 | p90 ribosomal S6 kinase inhibitor

    CAS:
    501437-28-1
    Catalog Number:
    10-4791
    Activity:
    p90 ribosomal S6 kinase inhibitor
    Chemical Name:
    2-(3,5-Difluoro-4-hydroxyanilino)-5,7-dimethyl-8-(3-methylbutyl)-7H-pteridin-6-one
    Molecular Weight:
    391.42
    Molecular Formula:
    C19H23F2N5O2
    Solubility:
    Soluble in DMSO (up to 15 mg/ml)
    Physical Properties:
    Off-white solid
    Purity:
    98%
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $90.00
    View Product This product has multiple variants. The options may be chosen on the product page
  • BX795 | Dual TBK1/IKKε inhibitor – enhances lentiviral transduction efficiency

    CAS:
    702675-74-9
    Catalog Number:
    10-4677
    Activity:
    Dual inhibitor of TBK1/IKKε
    Chemical Names:
    N-[3-[[5-Iodo-4-[3-(thiophene-2-carbonylamino)propylamino]pyrimidin-2-yl]amino]phenyl]pyrrolidine-1-carboxamide
    Molecular Weight:
    591.47
    Molecular Formula:
    C23H26IN7O2S
    Solubility:
    Soluble in DMSO (>25 mg/ml)
    Physical Properties:
    Off-white solid
    Purity:
    >97% HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $65.00
    View Product This product has multiple variants. The options may be chosen on the product page
  • Defactinib | Potent FAK inhibitor

    CAS:
    1073154-85-4
    Catalog Number:
    10-4828
    Activity:
    Potent FAK inhibitor
    Chemical Name:
    N-Methyl-4-[[4-[[3-[methyl(methylsulfonyl)amino]pyrazin-2-yl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]aminl]benzamide
    Molecular Weight:
    510.50
    Molecular Formula:
    C20H21F3N8O3S
    Solubility:
    Soluble in DMSO (up to at least 25mg/ml)
    Physical Properties:
    White solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C (des.)
    Stability:
    Stable for 1 year as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $65.00
    View Product This product has multiple variants. The options may be chosen on the product page
  • Deucravacitinib | Allosteric TYK2 inhibitor

    CAS:
    1609392-27-9
    Catalog Number:
    10-4756
    Activity:
    Allosteric TYK2 inhibitor
    Chemical Names:
    6-(Cyclopropanecarbonylamino)-4-[2-methoxy-3-(1-methyl-1,2,4-triazol-3-yl)anilino]-N-(trideuteriomethyl)pyridazine-3-carboxamide
    Alternate Name:
    BMS-986165
    Molecular Weight:
    425.47
    Molecular Formula:
    C20H19D3N8O3
    Solubility:
    Soluble in DMSO (25 mg/ml with warming); ethanol (20 mg/ml)
    Physical Properties:
    White to off-white solid
    Purity:
    >98% HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $100.00
    View Product This product has multiple variants. The options may be chosen on the product page
  • Duvelisib | PI3Kdelta/gamma inhibitor

    CAS:
    1201438-56-3
    Catalog Number:
    10-4788
    Activity:
    PI3Kδ/γ inhibitor/Cancer immunotherapy enhancer
    Chemical Name:
    8-Chloro-2-phenyl-3-[(1S)-1-(7H-purin-6-ylamino)ethyl]isoquinolin-1-one
    Alternative Name:
    IPI-145
    Molecular Weight:
    416.87
    Molecular Formula:
    C22H17ClN6O
    Solubility:
    Soluble in DMSO (up to at least 25 mg/ml)
    Physical Properties:
    White solid
    Purity:
    98% by HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $65.00
    View Product This product has multiple variants. The options may be chosen on the product page
1 2 3 4 5 6 7

20% OFF

For Postdoc
Customers!