Sodium channels

  • A-438079 HCl | P2X7 antagonist

    CAS:
    899431-18-6
    Catalog Number:
    10-4063
    Activity:
    P2X7 antagonist
    Chemical Names:
    3-[5-(2,3-Dichlorophenyl)tetrazol-1-ylmethyl]pyridine hydrochloride
    Molecular Weight:
    342.61
    Molecular Formula:
    C13H9Cl2N5·HCl
    Solubility:
    Soluble in DMSO (>25 mg/ml)
    Physical Properties:
    White to off-white solid
    Purity:
    >98% HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
    Shipping Code:
    RT
    From $60.00
  • A-803467 | NaV1.8 blocker

    CAS:
    944261-79-4
    Catalog Number:
    10-1066
    Activity:
    NaV1.8 blocker
    Chemical Name:
    5-(4-Chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-carboxamide
    Molecular Weight:
    357.8
    Molecular Formula:
    C19H16ClNO4
    Solubility:
    Soluble in DMSO (up to 15 mg/ml) or in Ethanol (up to 2 mg/ml).
    Physical Properties:
    White solid
    Purity:
    98% by TLC
    NMR (Conforms)
    Storage Temperature:
    RT
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $50.00
  • BAY-1797 | P2X4 antagonist

    CAS:
    2055602-83-8
    Catalog Number:
    10-3980
    Activity:
    P2X4 antagonist
    Chemical Names:
    N-[4-(3-Chlorophenoxy)-3-sulfamoylphenyl]-2-phenylacetamide
    Molecular Weight:
    416.88
    Molecular Formula:
    C20H17ClN2O4S
    Solubility:
    Soluble in DMSO (>25 mg/ml)
    Physical Properties:
    Pale brown solid
    Purity:
    >98% HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $75.00
  • ICA-121431 | Selective Sodium channel blocker

    CAS:
    313254-51-2
    Catalog Number:
    10-4085
    Activity:
    Selective Nav1.1/1.3 inhibitor
    Chemical Names:
    2,2-Diphenyl-N-[4-(1,3-thiazol-2-ylsulfamoyl)phenyl]acetamide
    Molecular Weight:
    449.54
    Molecular Formula:
    C23H19N3O3S2
    Solubility:
    Soluble in DMSO (>25 mg/ml)
    Physical Properties:
    Off-white to beige solid
    Purity:
    >98% TLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $50.00
  • PF-05089771 | Selective Nav1.7 inhibitor

    CAS:
    1235403-62-9
    Catalog Number:
    10-3990
    Activity:
    Selective Nav1.7 channel blocker
    Chemical Name:
    4-[2-(5-Amino-1H-pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide
    Alternate Name:
    PF771
    Molecular Weight:
    500.34
    Molecular Formula:
    C18H12Cl2FN5O3S2
    Solubility:
    Soluble in DMSO (>25 mg/ml)
    Physical Properties:
    White solid
    Purity:
    >98% HPLC
    NMR (Conforms)
    Storage Temperature:
    -20°C
    Stability:
    Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
    Shipping Code:
    RT
    From $60.00